HIV Citation List: February 18 - March 3, 2009

Pubmed citations:

1. Design, Synthesis and Anti-HIV Integrase Evaluation of 4-Oxo-4H-quinolizine-3-carboxylic Acid Derivatives. Xu YS, Zeng CC, Jiao ZG, Hu LM, Zhong RG. Molecules. 2009 Feb 19;14(2):868-83.

PMID: 19255545

2. Efficient inhibition of SDF-1alpha-mediated chemotaxis and HIV-1 infection by novel CXCR4 antagonists. Iwasaki Y, Akari H, Murakami T, Kumakura S, Dewan MZ, Yanaka M, Yamamoto N. Cancer Sci. 2009 Feb 23. [Epub ahead of print]

PMID: 19245436

3. Raltegravir: The First HIV Type 1 Integrase Inhibitor. Hicks C, Gulick RM. Clin Infect Dis. 2009 Feb 20. [Epub ahead of print]

PMID: 19231980

4. Design, synthesis, and biological evaluation of novel quinoline derivatives as HIV-1 Tat-TAR interaction inhibitors. Chen S, Chen R, He M, Pang R, Tan Z, Yang M. Bioorg Med Chem. 2009 Mar 1;17(5):1948-56. Epub 2009 Jan 23.

PMID: 19217787

5. 1-Amido-1-phenyl-3-piperidinylbutanes--CCR5 antagonists for the treatment of HIV: Part 2. Barber CG, Blakemore DC, Chiva JY, Eastwood RL, Middleton DS, Paradowski KA. Bioorg Med Chem Lett. 2009 Mar 1;19(5):1499-503. Epub 2009 Jan 10.

PMID: 19185490

6. GRL-02031, a novel nonpeptidic protease inhibitor (PI) containing a stereochemically defined fused cyclopentanyltetrahydrofuran potent against multi-PI-resistant human immunodeficiency virus type 1 in vitro. Koh Y, Das D, Leschenko S, Nakata H, Ogata-Aoki H, Amano M, Nakayama M, Ghosh AK, Mitsuya H. Antimicrob Agents Chemother. 2009 Mar;53(3):997-1006. Epub 2008 Oct 27.

PMID: 18955518

7. Synthesis of alkenyldiarylmethanes (ADAMs) containing benzo[d]isoxazole and oxazolidin-2-one rings, a new series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors. Deng BL, Zhao Y, Hartman TL, Watson K, Buckheit RW Jr, Pannecouque C, De Clercq E, Cushman M. Eur J Med Chem. 2009 Mar;44(3):1210-4. Epub 2008 Sep 19.

PMID: 18952324

8. Nebrodeolysin, a novel hemolytic protein from mushroom Pleurotus nebrodensis with apoptosis-inducing and anti-HIV-1 effects. Lv H, Kong Y, Yao Q, Zhang B, Leng FW, Bian HJ, Balzarini J, Van Damme E, Bao JK. Phytomedicine. 2009 Mar;16(2-3):198-205. Epub 2008 Aug 21.

PMID: 18722099

9. Synthesis and in vitro anti-HIV evaluation of a new series of 6-arylmethyl-substituted S-DABOs as potential non-nucleoside HIV-1 reverse transcriptase inhibitors. Wang YP, Chen FE, De Clercq E, Balzarini J, Pannecouque C. Eur J Med Chem. 2009 Mar;44(3):1016-23. Epub 2008 Jul 4.

PMID: 18692274

10. Design of Peptide-based Inhibitors for Human Immunodeficiency Virus Type 1 Strains Resistant to T-20. Izumi K, Kodama E, Shimura K, Sakagami Y, Watanabe K, Ito S, Watabe T, Terakawa Y, Nishikawa H, Sarafianos SG, Kitaura K, Oishi S, Fujii N, Matsuoka M. J Biol Chem. 2009 Feb 20;284(8):4914-20. Epub 2008 Dec 10.

PMID: 19073606

11. 5'-aminocarbonyl phosphonates as new zidovudine depot forms: antiviral properties, intracellular transformations, and pharmacokinetic parameters. Khandazhinskaya AL, Yanvarev DV, Jasko MV, Shipitsin AV, Khalizev VA, Shram SI, Skoblov YS, Shirokova EA, Kukhanova MK. Drug Metab Dispos. 2009 Mar;37(3):494-501. Epub 2008 Dec 23.

PMID: 19106116

12. A Trypsin-Chymotrypsin Inhibitor with Antiproliferative Activity from Small Glossy Black Soybeans. Ye X, Bun Ng T. Planta Med. 2009 Feb 20. [Epub ahead of print]

PMID: 19235124

13. Multivalent interactions with gp120 are required for the anti-HIV activity of cyanovirin. Liu Y, Carroll JR, Holt LA, Mc Mahon J, Giomarelli B, Ghirlanda G. Biopolymers. 2009 Feb 23. [Epub ahead of print]

PMID: 19235857

14. Lycojapodine A, a Novel Alkaloid from Lycopodium japonicum. He J, Chen XQ, Li MM, Zhao Y, Xu G, Cheng X, Peng LY, Xie MJ, Zheng YT, Wang YP, Zhao QS. Org Lett. 2009 Feb 26. [Epub ahead of print]

PMID: 19245240

15. Predicting anti-HIV activity of 1,3,4-thiazolidinone derivatives: 3D-QSAR approach. Ravichandran V, Prashantha Kumar BR, Sankar S, Agrawal RK. Eur J Med Chem. 2009 Mar;44(3):1180-7. Epub 2008 Jun 12.

PMID: 18687505

ISI Web of Science citations:

16. Investigation on the role of the tetrazole in the binding of thiotetrazolylacetanilides with HIV-1 wild type and K103N/Y181C double mutant reverse transcriptases. Gagnon A, Landry S, Coulombe R, Jakalian A, Guse I, Thavonekham B, Bonneau PR, Yoakim C, Simoneau B. SO BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2009;19(4):1199-1205

17. Synthesis of 5-isoxazol-5-yl-2 '-deoxyuridines exhibiting antiviral activity against HSV and several RNA viruses. Lee YS, Park SM, Kim BH. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2009;19(4):1126-1128.

18. Synthesis of Zidovudine Derivatives with Anti-HIV-1 and Antibacterial Activities. Senthilkumar P, Long J, Swetha R, Shruthi V, Wang RR, Preethi S, Yogeeswari P, Zheng YT, Sriram D. NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS. 2009;28(2):89-102.

19. A facile synthesis of 2,3-disubstituted furo[2,3-b]pyridines. Beutner GL, Kuethe JT, Yasuda N. TETRAHEDRON LETTERS. 2009;50(7):781-784.

20. A novel and efficient synthesis of chiral C-2-symmetric 1,4-diamines. Xu LH, Desai MC, Liu HT. TETRAHEDRON LETTERS. 2009;50(5):552-554.

21. Routes to HIV-integrase inhibitors: efficient synthesis of bicyclic pyrimidones by ring expansion or amination at a benzylic position. Ferreira MDR, Cecere G, Pace P, Summa V. TETRAHEDRON LETTERS. 2009;50(2):148-151.

22. BIOLOGICAL ACTIVITY OF METHYL 2-[5-OXO-3,4-DI-(2-PIRYDYL)-1,4,5,6-TETRAHYDRO-1,2,4-TRIAZINE-6-YLIDENE] ACETATE. Ucherek MM, Wroblewska J, Modzelewska-Banachiewicz B, Gospodarek E. ACTA POLONIAE PHARMACEUTICA. 2008;65(6):789-791.

23. Sidechain-linked inhibitors of HIV-1 protease dimerization. Bowman MJ, Chmielewski J. BIOORGANIC & MEDICINAL CHEMISTRY. 2009;17(3):967-976.

24. Ring-Opening Polymerization of Benzylated 1,6-Anhydro-beta-D-lactose and Specific Biological Activities of Sulfated (1 -> 6)-alpha-D-Lactopyranans. Han S, Kanematsu Y, Hattori K, Nakashima H, Yoshida T. JOURNAL OF POLYMER SCIENCE PART A-POLYMER CHEMISTRY. 2009;47(3):913-924.

25. A New Strategy for the Synthesis of Optically Pure beta-Fluoroalkyl beta-Amino Acid Derivatives. Fustero S, del Pozo C, Catalan S, Aleman J, Parra A, Marcos V, Ruano JLG. ORGANIC LETTERS. 2009;11(3):641-644.

26. Polymethylene derivatives of nucleic bases with omega-functional groups: VII. Cytotoxicity in the series of N-(2-oxocyclohexyl)-omega-oxoalkyl-substituted purines and pyrimidines. Komissarov VV, Volgareva GM, Ol'shanskaya YS, Chernyshova ME, Zavalishina LE, Frank GA, Shtil' AA, Kritzyn AM. RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY. 2009;35(1):75-85.

27. Synthesis and Antiviral Evaluation of (-)-3 '-Methylcarbovir, (-)-3 '-Methylabacavir, and Modified Purine Analogues. Bremond P, Audran G, Monti H, De Clercq E, Pannecouque C. SYNTHESIS-STUTTGART. 2009;2:290-296.