HIV Citation List: December 25 - January 6, 2009

Anti*HIV

1. Anti Human Immunodeficiency Virus-1 (HIV-1) Agents 1. Discovery of Benzyl Phenyl Ethers as New HIV-1 Inhibitors in Vitro.

Dai HL, Liu WQ, Xu H, Yang LM, Lv M, Zheng YT.

Chem Pharm Bull (Tokyo). 2009 Jan;57(1):84-6.

PMID: 19122322 [PubMed - in process]

2. High-throughput screening using pseudotyped lentiviral particles: A strategy for the identification of HIV-1 inhibitors in a cell-based assay.

Garcia JM, Gao A, He PL, Choi J, Tang W, Bruzzone R, Schwartz O, Naya H, Nan FJ, Li J, Altmeyer R, Zuo JP.

Antiviral Res. 2008 Dec 29. [Epub ahead of print]

PMID: 19118579 [PubMed - as supplied by publisher]

3. Design, synthesis, and biological evaluation of N-carboxyphenylpyrrole derivatives as potent HIV fusion inhibitors targeting gp41.

Liu K, Lu H, Hou L, Qi Z, Teixeira C, Barbault F, Fan BT, Liu S, Jiang S, Xie L.

J Med Chem. 2008 Dec 25;51(24):7843-54.

PMID: 19053778 [PubMed - in process]

4. Development and preclinical studies of broad-spectrum anti-HIV agent (3'R,4'R)-3-cyanomethyl-4-methyl-3',4'-di-O-(S)-camphanoyl-(+)-cis-khellactone (3-cyanomethyl-4-methyl-DCK).

Xie L, Guo HF, Lu H, Zhuang XM, Zhang AM, Wu G, Ruan JX, Zhou T, Yu D, Qian K, Lee KH, Jiang S.

J Med Chem. 2008 Dec 25;51(24):7689-96.

PMID: 19053755 [PubMed - in process]

5. Novel nucleotide human immunodeficiency virus reverse transcriptase inhibitor GS-9148 with a low nephrotoxic potential: characterization of renal transport and accumulation.

Cihlar T, Laflamme G, Fisher R, Carey AC, Vela JE, Mackman R, Ray AS.

Antimicrob Agents Chemother. 2009 Jan;53(1):150-6. Epub 2008 Nov 10.

PMID: 19001108 [PubMed - in process]

6. Synthesis, HIV-RT inhibitory activity and SAR of 1-benzyl-1H-1,2,3-triazole derivatives of carbohydrates.

da Silva Fde C, de Souza MC, Frugulhetti II, Castro HC, Souza SL, de Souza TM, Rodrigues DQ, Souza AM, Abreu PA, Passamani F, Rodrigues CR, Ferreira VF.

Eur J Med Chem. 2009 Jan;44(1):373-83. Epub 2008 Mar 16.

PMID: 18486994 [PubMed - in process]

7. Synthesis and anti-HIV-1 integrase activities of 3-aroyl-2,3-dihydro-1,1-dioxo-1,4,2-benzodithiazines.

Brzozowski Z, Saczewski F, Sławiński J, Sanchez T, Neamati N.

Eur J Med Chem. 2009 Jan;44(1):190-6. Epub 2008 Mar 4.

PMID: 18394758 [PubMed - in process]

Compound and (HIV or AIDS or Human Immunodeficiency Virus)

8. Cyanovirin-N potently inhibits human immunodeficiency virus type 1 infection in cellular and cervical explant models.

Buffa V, Stieh D, Mamhood N, Hu Q, Fletcher P, Shattock RJ.

J Gen Virol. 2009 Jan;90(Pt 1):234-43.

PMID: 19088294 [PubMed - in process]

9. Inhibition of human immunodeficiency virus (HIV-1) infection in human peripheral blood leucocytes-SCID reconstituted mice by rapamycin.

Nicoletti F, Lamenta C, Donati S, Spada M, Ranazzi A, Cacopardo B, Mangano K, Belardelli F, Perno C, Aquaro S.

Clin Exp Immunol. 2009 Jan;155(1):28-34.

PMID: 19076826 [PubMed - in process]

10. Synthesis and in vitro activities of a new antiviral duplex drug linking Zidovudine (AZT) and Foscarnet (PFA) via an octadecylglycerol residue.

Schott H, Hamprecht K, Schott S, Schott TC, Schwendener RA.

Bioorg Med Chem. 2009 Jan 1;17(1):303-10. Epub 2008 Nov 5.

PMID: 19010684 [PubMed - in process]

11. Non-nucleoside HIV-1 reverse transcriptase inhibitors di-halo-indolyl aryl sulfones achieve tight binding to drug-resistant mutants by targeting the enzyme-substrate complex.

Samuele A, Kataropoulou A, Viola M, Zanoli S, La Regina G, Piscitelli F, Silvestri R, Maga G.

Antiviral Res. 2009 Jan;81(1):47-55. Epub 2008 Nov 5.

PMID: 18984007 [PubMed - in process]

12. A New Generation of Peptide-based Inhibitors Targeting HIV-1 Reverse Transcriptase Conformational Flexibility.

Agopian A, Gros E, Aldrian-Herrada G, Bosquet N, Clayette P, Divita G.

J Biol Chem. 2009 Jan 2;284(1):254-64. Epub 2008 Oct 23.

PMID: 18952602 [PubMed - in process]

Inhibition and (HIV or AIDS or Human Immunodeficiency Virus)

13. SC29EK, a peptide fusion inhibitor with enhanced {alpha}-helicity, inhibits replication of human immunodeficiency virus type 1 mutants resistant to enfuvirtide.

Naito T, Izumi K, Kodama E, Sakagami Y, Kajiwara K, Nishikawa H, Watanabe K, Sarafianos SG, Oishi S, Fujii N, Matsuoka M.

Antimicrob Agents Chemother. 2008 Dec 29. [Epub ahead of print]

PMID: 19114674 [PubMed - as supplied by publisher]

14. Complete absolute configuration of integramide A, a natural, 16-mer peptide inhibitor of HIV-1 integrase, elucidated by total synthesis.

De Zotti M, Formaggio F, Kaptein B, Broxterman QB, Felock PJ, Hazuda DJ, Singh SB, Brückner H, Toniolo C.

Chembiochem. 2009 Jan 5;10(1):87-90. No abstract available.

PMID: 18850604 [PubMed - in process]

Citations From The Forwarded 'Web of Knowledge' listings

15. Design of Annulated Pyrazoles as Inhibitors of HIV-1 Reverse Transcriptase.

Sweeney ZK, Harris SF, Arora N, Javanbakht H, Li Y, Fretland J, Davidson JP, Billedeau JR, Gleason SK, Hirschfeld D, Kennedy-Smith JJ, Mirzadegan T, Roetz R, Smith M, Sperry S, Suh JM, Wu J, Tsing S, Villaseñor AG, Paul A, Su G, Heilek G, Hang JQ, Zhou AS, Jernelius JA, Zhang FJ, Klumpp K.

J Med Chem. 2008 Nov 14. [Epub ahead of print]

PMID: 19007201 [PubMed - as supplied by publisher]

16. Synthesis and Bioactivity of Dibenzylbutance Ligans and Their Anaologues

Xia YM, Bi WH and Cao XP

Chemical Journal of Chinese Universities. 2008 Nov; 29(11): 2178-2182.

17. Optimization of 5-aryloxyimidazole non-nucleoside reverse transcriptase inhibitors.

Jones LH, Allan G, Corbau R, Hay D, Middleton DS, Mowbray CE, Newman SD, Perros M, Randall A, Vuong H, Webster R, Westby M, Williams D.

ChemMedChem. 2008 Nov;3(11):1756-62.

PMID: 18855969 [PubMed - in process]

18. Synthesis and Anti-HIV-1 Activity of Carbocyclic Versions of Stavudine Analogues using a Ring-Closing Metathesis

Liu LJ, Ko OH and Hong JH

Bulletin of the Korean Chemical Society. 2008 Sep; 29(9): 1723-28.

19. Marmorin, a new ribosome inactivating protein with antiproliferative and HIV-1 reverse transcriptase inhibitory activities from the mushroom Hypsizigus marmoreus.

Wong JH, Wang HX, Ng TB.

Appl Microbiol Biotechnol. 2008 Dec;81(4):669-74. Epub 2008 Aug 27.

PMID: 18751697 [PubMed - in process]