HIV Citation List: October 30 - November 12, 2008
Anti-HIV
1. Hunter R, Younis Y, Muhanji CI, Curtin TL, Naidoo KJ, Petersen M, Bailey CM, Basavapathruni A, Anderson KS.
C-2-Aryl O-substituted HI-236 derivatives as non-nucleoside HIV-1 reverse-transcriptase inhibitors.
Bioorg Med Chem. 2008 Nov 1. [Epub ahead of print]
PMID: 18996020 [PubMed - as supplied by publisher]
2. Ghosh SK, Patra R, Rath SP.
Axial ligand coordination in sterically strained vanadyl porphyrins: synthesis, structure, and properties.
Inorg Chem. 2008 Nov 3;47(21):9848-56. Epub 2008 Sep 30.
PMID: 18823111 [PubMed - in process]
3. Qi Z, Shi W, Xue N, Pan C, Jing W, Liu K, Jiang S.
Rationally Designed Anti-HIV Peptides Containing Multifunctional Domains as Molecule Probes for Studying the Mechanisms of Action of the First and Second Generation HIV Fusion Inhibitors.
J Biol Chem. 2008 Oct 31;283(44):30376-84. Epub 2008 Jul 28.
PMID: 18662985 [PubMed - in process]
Anti-Viral and HIV
4. Cohen C, Forzan M, Sproat B, Pantophlet R, McGowan I, Burton D, James W.
An aptamer that neutralizes R5 strains of HIV-1 binds to core residues of gp120 in the CCR5 binding site.
Virology. 2008 Nov 10;381(1):46-54. Epub 2008 Sep 17.
PMID: 18799178 [PubMed - in process]
(HIV or AIDS) and (Therapeutic or Compound)
5. Samuele A, Kataropoulou A, Viola M, Zanoli S, La Regina G, Piscitelli F, Silvestri R, Maga G.
Non-nucleoside HIV-1 reverse transcriptase inhibitors di-halo-indolyl aryl sulfones achieve tight binding to drug-resistant mutants by targeting the enzyme-substrate complex.
Antiviral Res. 2008 Nov 1. [Epub ahead of print]
PMID: 18984007 [PubMed - as supplied by publisher]
6. Van Neck T, Pannecouque C, Vanstreels E, Stevens M, Dehaen W, Daelemans D.
Inhibition of the CRM1-mediated nucleocytoplasmic transport by N-azolylacrylates: structure-activity relationship and mechanism of action.
Bioorg Med Chem. 2008 Nov 1;16(21):9487-97. Epub 2008 Sep 20.
PMID: 18835718 [PubMed - in process]
7. Sapre NS, Gupta S, Pancholi N, Sapre N.
Data mining using template-based molecular docking on tetrahydroimidazo-[4,5,1-jk][1,4]-benzodiazepinone (TIBO) derivatives as HIV-1RT inhibitors.
J Mol Model. 2008 Nov;14(11):1009-21. Epub 2008 Jul 19.
PMID: 18642033 [PubMed - in process]
(HIV or AIDS) and Inhibition
8. Michalowski D, Chitima-Matsiga R, Held DM, Burke DH.
Novel bimodular DNA aptamers with guanosine quadruplexes inhibit phylogenetically diverse HIV-1 reverse transcriptases.
Nucleic Acids Res. 2008 Nov 7. [Epub ahead of print]
PMID: 18996899 [PubMed - as supplied by publisher]
9. Bacchi A, Biemmi M, Carcelli M, Carta F, Compari C, Fisicaro E, Rogolino D, Sechi M, Sippel M, Sotriffer CA, Sanchez TW, Neamati N.
From Ligand to Complexes. Part 2. Remarks on Human Immunodeficiency Virus type 1 Integrase Inhibition by beta-Diketo Acid Metal Complexes.
J Med Chem. 2008 Nov 5. [Epub ahead of print]
PMID: 18983138 [PubMed - as supplied by publisher]
10. Van Neck T, Pannecouque C, Vanstreels E, Stevens M, Dehaen W, Daelemans D.
Inhibition of the CRM1-mediated nucleocytoplasmic transport by N-azolylacrylates: structure-activity relationship and mechanism of action.
Bioorg Med Chem. 2008 Nov 1;16(21):9487-97. Epub 2008 Sep 20.
PMID: 18835718 [PubMed - in process]
(HIV or AIDS) and Inhibitor
11. Elworthy TR, Dunn JP, Hogg JH, Lam G, Saito YD, Silva TM, Stefanidis D, Woroniecki W, Zhornisky E, Zhou AS, Klumpp K.
Orally bioavailable prodrugs of a BCS class 2 molecule, an inhibitor of HIV-1 reverse transcriptase.
Bioorg Med Chem Lett. 2008 Nov 1. [Epub ahead of print]
PMID: 18993071 [PubMed - as supplied by publisher]
(HIV or AIDS) and (Therapeutic or Compound or Pharmaceutical)
12. Asamitsu K, Yamaguchi T, Nakata K, Hibi Y, Victoriano AF, Imai K, Onozaki K, Kitade Y, Okamoto T.
Inhibition of Human Immunodeficiency Virus Type 1 Replication by Blocking I{kappa}B Kinase with Noraristeromycin.
J Biochem. 2008 Nov;144(5):581-589. Epub 2008 Aug 19.
PMID: 18713798 [PubMed - as supplied by publisher]
Journal Check
13. Radi M, Angeli L, Franchi L, Contemori L, Maga G, Samuele A, Zanoli S, Armand-Ugon M, Gonzalez E, Llano A, Esté JA, Botta M.
Towards novel S-DABOC inhibitors: Synthesis, biological investigation, and molecular modeling studies.
Bioorg Med Chem Lett. 2008 Sep 23. [Epub ahead of print]
PMID: 18842407 [PubMed - as supplied by publisher]
14. Maga G, Falchi F, Garbelli A, Belfiore A, Witvrouw M, Manetti F, Botta M.
Pharmacophore modeling and molecular docking led to the discovery of inhibitors of human immunodeficiency virus-1 replication targeting the human cellular aspartic acid-glutamic acid-alanine-aspartic acid box polypeptide 3.
J Med Chem. 2008 Nov 13;51(21):6635-8. Epub 2008 Oct 4.
PMID: 18834110 [PubMed - in process]