ONLINE DATABASE SEARCH - HIV-LS-361-MEMO
1. 59375 HIV-LS-361; PUBMED-HIV-11/13/2006
Synthesis and anti-HIV activity evaluation of 1-[(alkenyl or alkynyl or alkyloxy)methyl]-5-alkyl-6-(1-naphthoyl)-2,4-pyrimidinediones as novel non-nucleoside HIV-1 reverse transcriptase inhibitors
Ji, L, Chen, FE, Xie, B, De, Clercq E, Balzarini, J, and Pannecouque, C
Eur J Med Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17095124&dopt=abstract
2. 59376 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Preparation of bicyclic heterocycles, particularly pyrimido[2,1-c][1,4]oxazine-2-carboxamides, as HIV integrase inhibitors
Naidu, BNarasimhulu, Banville, Jacques, Beaulieu, Francis, Connolly, Timothy P, Krystal, Mark R, Matiskella, John D, Ouellet, Carl, Plamondon, Serge, Remillard, Roger, Sorenson, Margaret E, Ueda, Yasutsugu, and Walker, Michael A
PATENT: US 2006199956 ISSUE DATE: 20060907
APPLICATION: 2005-26389 PP: 182pp., Cont.-in-part of U.S. Ser. No. 126,891.
ASSIGNEE: (USA)
3. 59377 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Anti-HIV quinuclidine compounds
Lecanu, Laurent, Greeson, Janet, and Papadopoulos, Vassilios
PATENT: WO 2006085890 ISSUE DATE: 20060817
APPLICATION: 2005 PP: 28pp.
ASSIGNEE: (Samaritan Pharmaceuticals, Inc. USA and Georgetown University)
4. 59378 HIV-LS-361; PUBMED-HIV-11/13/2006
Anti-HIV-1 Constituents from Leaves and Twigs of Cratoxylum arborescens
Reutrakul, V, Chanakul, W, Pohmakotr, M, Jaipetch, T, Yoosook, C, Kasisit, J, Napaswat, C, Santisuk, T, Prabpai, S, Kongsaeree, P, and Tuchinda, P
Planta Med 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17091434&dopt=abstract
5. 59379 HIV-LS-361; PUBMED-HIV-11/13/2006
Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis, Structure-Activity Relationships, and Docking Studies (Part 2)
Lavecchia, A, Costi, R, Artico, M, Miele, G, Novellino, E, Bergamini, A, Crespan, E, Maga, G, and Di, Santo R
ChemMedChem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17089434&dopt=abstract
6. 59380 HIV-LS-361; PUBMED-HIV-11/13/2006
Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis, Structure-Activity Relationships, and Docking Studies (Part 1)
Di Santo, R, Costi, R, Artico, M, Miele, G, Lavecchia, A, Novellino, E, Bergamini, A, Cancio, R, and Maga, G
ChemMedChem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17089433&dopt=abstract
7. 59381 HIV-LS-361; PUBMED-HIV-11/13/2006
Molecular Mechanism by which K70E in HIV-1 Reverse Transcriptase Confers Resistance to Nucleoside Reverse Transcriptase Inhibitors
Sluis-Cremer, N, Sheen, CW, Zelina, S, Argoti, Torres PS, Parikh, UM, and Mellors, JW
Antimicrob Agents Chemother 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17088490&dopt=abstract
8. 59382 HIV-LS-361; PUBMED-HIV-11/13/2006
Critical role of the N-loop and beta1-strand hydrophobic clusters of RANTES-derived peptides in anti-HIV activity
Vangelista, L, Longhi, R, Sironi, F, Pavone, V, and Lusso, P
Biochem Biophys Res Commun 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17083916&dopt=abstract
9. 59383 HIV-LS-361; PUBMED-HIV-11/13/2006
The Role of V1V2 and other HIV-1 Envelope Domains in Resistance to Autologous Neutralization during Clade C Infection
Rong, R, Bibollet-Ruche, F, Mulenga, J, Allen, S, Blackwell, JL, and Derdeyn, CA
J Virol 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17079307&dopt=abstract
10. 59384 HIV-LS-361; PUBMED-HIV-11/13/2006
Ring substituent effects on biological activity of vinyl sulfones as inhibitors of HIV-1
Meadows, DC, Sanchez, T, Neamati, N, North, TW, and Gervay-Hague, J
Bioorg Med Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17074494&dopt=abstract
11. 59385 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Discovery, synthesis and optimization of a new series of selective HIV integrase inhibitors leading to MK-0518 currently in Phase III clinical trial for treatment of HIV/AIDS
Summa, Vincenzo
Abstracts of Papers, 232nd ACS National Meeting, San Francisco, CA, United States, Sept. 10-14, 2006 2006.: MEDI-298
12. 59386 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Short-term antiviral activity of TMC278 - a novel NNRTI - in treatment-naive HIV-1-infected subjects
Goebel, Frank, Yakovlev, Alexy, Pozniak, Anton L, Vinogradova, Elena, Boogaerts, Griet, Hoetelmans, Richard, de Bethune, Marie-Pierre P, Peeters, Monika, and Woodfall, Brian
AIDS (Hagerstown, MD, United States) 2006. 20(13): 1721-1726
13. 59387 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Rational design of polymerase inhibitors as antiviral drugs
Oeberg, Bo
Antiviral Research 2006. 71(2-3): 90-95
14. 59388 HIV-LS-361; SCIFINDER-HIV-11/7/2006
CoMFA study on quinolones as novel inhibitors of HIV-1 reverse transcriptase
Yi, Ping and Qiu, Minghua
Jisuanji Yu Yingyong Huaxue 2006. 23(5): 399-402
15. 59389 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Synthesis, antiviral and cytotoxicity of some new sulphonamides
Selvam, P, Abileshini, B, Alagarsamy, V, Pannecouque, C, and De Clercq, E
Indian Journal of Heterocyclic Chemistry 2006. 16(1): 73-74
16. 59390 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Phosphonate analogs of hiv inhibitor compounds
Boojamra, Constantine G, Lin, Kuei-Ying, Mackman, Richard L, Markevitch, David Y, Petrakovsky, Oleg V, Ray, Adrian S, and Zhang, Lijun
PATENT: WO 2006110157 ISSUE DATE: 20061019
APPLICATION: 2005 PP: 511pp.
ASSIGNEE: (Gilead Sciences, Inc. USA
17. 59391 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Suppression of HIV-1 Protease Inhibitor Resistance by Phosphonate-mediated Solvent Anchoring
Cihlar, Tomas, He, Gong-Xin, Liu, Xiaohong, Chen, James M, Hatada, Marcos, Swaminathan, Swami, McDermott, Martin J, Yang, Zheng-Yu, Mulato, Andrew S, Chen, Xiaowu, Leavitt, Stephanie A, Stray, Kirsten M, and Lee, William A
Journal of Molecular Biology 2006. 363(3): 635-647
18. 59392 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Fused pyrimidinones as HIV integrase inhibitors and their preparation and use in the treatment of HIV infection
Cecere, Giuseppe, Ferreira, Maria Del Rosario Rico, Jones, Philip, Pace, Paola, Petrocchi, Alessia, and Summa, Vincenzo
PATENT: WO 2006103399 ISSUE DATE: 20061005
APPLICATION: 2006 PP: 163pp.
ASSIGNEE: (Istituto De Ricerche Di Biologia Molecolare P Angeletti SpA, Italy
19. 59393 HIV-LS-361; SCIFINDER-HIV-11/7/2006
Fatty acid conjugates with HIV gp41-derived peptide for treatment of HIV infections
Wring, Stephen, Frick, Lloyd, Schneider, Stephen, Zhang, Huyi, Di, Jie, and Heilman, David
PATENT: WO 2006105201 ISSUE DATE: 20061005
APPLICATION: 2006 PP: 118pp.
ASSIGNEE: (Trimeris, Inc. USA
20. 59394 HIV-LS-361; WOS-HIV-11/6/2006
Solution structures and characterization of human immunodeficiency virus Rev responsive element IIB RNA targeting zinc finger proteins
Mishra, SH, Shelley, CM, Barrow, DJ, Darby, MK, and Germann, MW
BIOPOLYMERS 2006. 83(4): 352-364, 13
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000241344000003
21. 59395 HIV-LS-361; WOS-HIV-11/13/2006
The engagement of activating Fc gamma Rs inhibits primate lentivirus replication in human macrophages
David, A, Saez-Cirion, A, Versmisse, P, Malbec, O, Iannascoli, B, Herschke, F, Lucas, M, Barre-Sinoussi, F, Mouscadet, JF, Daeron, M, and Pancino, G
JOURNAL OF IMMUNOLOGY 2006. 177(9): 6291-6300, 10
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000241477400063