ONLINE DATABASE SEARCH -HIV-LS-344-MEMO
1. 48605 HIV-LS-344; PUBMED-HIV-3/20/2006
The effect of a methyl or 2-fluoroethyl substituent at the N-3 position of thymidine, 3'-fluoro-3'-deoxythymidine and 1-beta-D-arabinosylthymine on their antiviral and cytostatic activity in cell culture
Balzarini, J, Celen, S, Karlsson, A, de Groot, T, Verbruggen, A, and Bormans, G
Antivir Chem Chemother 2006. 17(1): 17-23
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16542002&dopt=abstract
2. 48606 HIV-LS-344; PUBMED-HIV-3/20/2006
Inhibition of HIV-1 replication by oligonucleotide analogues directed to the packaging signal and trans-activating response region
Brown, DE, Arzumanov, A, Syed, S, Gait, MJ, and Lever, AM
Antivir Chem Chemother 2006. 17(1): 1-9
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16542000&dopt=abstract
3. 48607 HIV-LS-344; PUBMED-HIV-3/20/2006
Highly Potent and Orally Active CCR5 Antagonists as Anti-HIV-1 Agents: Synthesis and Biological Activities of 1-Benzazocine Derivatives Containing a Sulfoxide Moiety
Seto, M, Aikawa, K, Miyamoto, N, Aramaki, Y, Kanzaki, N, Takashima, K, Kuze, Y, Iizawa, Y, Baba, M, and Shiraishi, M
J Med Chem 2006. 49(6): 2037-2048
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16539392&dopt=abstract
4. 48608 HIV-LS-344; PUBMED-HIV-3/20/2006
Novel Bifunctional Quinolonyl Diketo Acid Derivatives as HIV-1 Integrase Inhibitors: Design, Synthesis, Biological Activities, and Mechanism of Action
Di Santo, R, Costi, R, Roux, A, Artico, M, Lavecchia, A, Marinelli, L, Novellino, E, Palmisano, L, Andreotti, M, Amici, R, Galluzzo, CM, Nencioni, L, Palamara, AT, Pommier, Y, and Marchand, C
J Med Chem 2006. 49(6): 1939-1945
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16539381&dopt=abstract
5. 48609 HIV-LS-344; EMBASE-HIV-3/20/2006
Inhibition of HIV entry by carbohydrate-binding proteins
Balzarini, J
Antiviral Research 2006. In Press, Uncorrected Proof
HYPERLINK:
http://www.sciencedirect.com/science/article/B6T2H-4JF8G1R-1/2/60befe4b223aa7be66ed1d6de0c3e6bf
6. 48610 HIV-LS-344; PUBMED-HIV-3/20/2006
New HIV-1 reverse transcriptase inhibitors based on a tricyclic benzothiophene scaffold: Synthesis, resolution, and inhibitory activity
Krajewski, K, Zhang, Y, Parrish, D, Deschamps, J, Roller, PP, and Pathak, VK
Bioorg Med Chem Lett 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16527484&dopt=abstract
7. 48611 HIV-LS-344; PUBMED-HIV-3/20/2006
A fluorescence polarization assay for screening inhibitors against the ribonuclease H activity of HIV-1 reverse transcriptase
Nakayama, GR, Bingham, P, Tan, D, and Maegley, KA
Anal Biochem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16527235&dopt=abstract
8. 48612 HIV-LS-344; PUBMED-HIV-3/20/2006
Design, synthesis, and biological evaluation of chicoric acid analogs as inhibitors of HIV-1 integrase
Charvat, TT, Lee, DJ, Robinson, WE, and Chamberlin, AR
Bioorg Med Chem 2006.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16524737&dopt=abstract
9. 48613 HIV-LS-344; PUBMED-HIV-3/20/2006
Structure-activity relationships of anti-HIV-1 peptides with disulfide linkage between D- and L-cysteine at positions i and i+3, respectively, derived from HIV-1 gp41 C-peptide
Lee, MK, Kim, HK, Lee, TY, Hahm, KS, and Kim, KL
Exp Mol Med 2006. 38(1): 18-26
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16520549&dopt=abstract
10. 48614 HIV-LS-344; EMBASE-HIV-3/20/2006
The HIV-1 reverse transcriptase mutants G190S and G190A, which confer resistance to non-nucleoside reverse transcriptase inhibitors, demonstrate reductions in RNase H activity and DNA synthesis from tRNALys, 3 that correlate with reductions in replication efficiency
Wang, J, Dykes, C, Domaoal, RA, Koval, CE, Bambara, RA, and Demeter, LM
Virology 2006. In Press, Corrected Proof
HYPERLINK:
http://www.sciencedirect.com/science/article/B6WXR-4JCBN4M-2/2/a604d73efcfd26101a6d40d48f6e92d4
11. 48615 HIV-LS-344; PUBMED-HIV-3/20/2006
Antiviral properties of two trimeric recombinant gp41 proteins
Delcroix-Genete, D, Quan, PL, Roger, MG, Hazan, U, Nisole, S, and Rousseau, C
Retrovirology 2006. 3(1): 16
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16515685&dopt=abstract
12. 48616 HIV-LS-344; PUBMED-HIV-3/20/2006
Dynamic pharmacophore model optimization: identification of novel HIV-1 integrase inhibitors
Deng, J, Sanchez, T, Neamati, N, and Briggs, JM
J Med Chem 2006. 49(5): 1684-92
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16509584&dopt=abstract
13. 48617 HIV-LS-344; PUBMED-HIV-3/20/2006
Synthesis and anti-HIV-1 and anti-HCMV activity of 1-substituted 3-(3,5-dimethylbenzyl)uracil derivatives
Maruyama, T, Kozai, S, Demizu, Y, Witvrouw, M, Pannecouque, C, Balzarini, J, Snoecks, R, Andrei, G, and De, Clercq E
Chem Pharm Bull (Tokyo) 2006. 54(3): 325-33
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16508186&dopt=abstract
14. 48618 HIV-LS-344; PUBMED-HIV-3/20/2006
Rubriflordilactones a and B, two novel bisnortriterpenoids from schisandrarubriflora and their biological activities
Xiao, WL, Yang, LM, Gong, NB, Wu, L, Wang, RR, Pu, JX, Li, XL, Huang, SX, Zheng, YT, Li, RT, Lu, Y, Zheng, QT, and Sun, HD
Org Lett 2006. 8(5): 991-4
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16494492&dopt=abstract
15. 48619 HIV-LS-344; WOS-HIV-3/12/2006
Dexelvucitabine - Anti-HIV agent - Reverse transcriptase inhibitor
McIntyre, JA and Castaner, J
DRUGS OF THE FUTURE 2005. 30(12): 1205-1211, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000235583600001
16. 48620 HIV-LS-344; WOS-HIV-3/12/2006
Discovery of a highly potent and orally active CCR5 antagonist TAK-652 as an anti-HIV-1 agent: Synthesis and biological activities of 1-benzazocine derivatives containing a sulfoxide moiety
Seto, M, Aikawa, K, Aramaki, Y, Miyamoto, N, Kanzaki, N, Kuze, Y, Takashima, K, Baba, M, and Shiraishi, M
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 2005. 229: U122-1
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000235066600088
17. 48621 HIV-LS-344; WOS-HIV-3/12/2006
Prodrugs of 1-(beta-d-dioxolane)thymine (DOT): Synthesis, anti-HIV-1 activity and stability study
Liang, YZ, Yadav, V, Schinazi, RF, and Chu, CK
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 2005. 229: U168-1
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000235066600333
18. 48622 HIV-LS-344; WOS-HIV-3/19/2006
In vitro development of resistance to human immunodeficiency virus protease inhibitor GW640385
Yates, PJ, Hazen, R, St, Clair M, Boone, L, Tisdale, M, and Elston, RC
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY 2006. 50(3): 1092-1095, 4
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000235786300039