ONLINE DATABASE SEARCH - HIV-LS-337-MEMO
1. 48219 HIV-LS-337; PUBMED-HIV-12/12/2005
Effect of a Bound Non-Nucleoside RT Inhibitor on the Dynamics of Wild-Type and Mutant HIV-1 Reverse Transcriptase
Zhou, Z, Madrid, M, Evanseck, JD, and Madura, JD
J Am Chem Soc 2005. 127(49): 17253-17260
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16332074&dopt=abstract
2. 48220 HIV-LS-337; PUBMED-HIV-12/12/2005
Synthesis and antiviral activities of 1,2,3-triazole functionalized thymidines: 1,3-dipolar cycloaddition for efficient regioselective diversity generation
Zhou, L, Amer, A, Korn, M, Burda, R, Balzarini, J, De Clercq, E, Kern, ER, and Torrence, PF
Antivir Chem Chemother 2005. 16(6): 375-383
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16331842&dopt=abstract
3. 48221 HIV-LS-337; PUBMED-HIV-12/12/2005
A novel small molecular weight compound with a carbazole structure that demonstrates potent human immunodeficiency virus type-1 integrase inhibitory activity
Yan, H, Mizutani, TC, Nomura, N, Takakura, T, Kitamura, Y, Miura, H, Nishizawa, M, Tatsumi, M, Yamamoto, N, and Sugiura, W
Antivir Chem Chemother 2005. 16(6): 363-73
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16329284&dopt=abstract
4. 48222 HIV-LS-337; PUBMED-HIV-12/12/2005
Synthesis and anti-HIV activity of new alkenyldiarylmethane (ADAM) non-nucleoside reverse transcriptase inhibitors (NNRTIs) incorporating benzoxazolone and benzisoxazole rings
Deng, BL, Cullen, MD, Zhou, Z, Hartman, TL, Buckheit, RW Jr, Pannecouque, C, Clercq, ED, Fanwick, PE, and Cushman, M
Bioorg Med Chem 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16321539&dopt=abstract
5. 48223 HIV-LS-337; PUBMED-HIV-12/12/2005
Dendritic Catanionic Assemblies: In vitro Anti-HIV Activity of Phosphorus-Containing Dendrimers Bearing Galbeta(1)cer Analogues
Blanzat, M, Turrin, CO, Aubertin, AM, Couturier-Vidal, C, Caminade, AM, Majoral, JP, Rico-Lattes, I, and Lattes, A
Chembiochem 2005. 6(12): 2207-2213
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16317767&dopt=abstract
6. 48224 HIV-LS-337; PUBMED-HIV-12/12/2005
Phosphoramidate and phosphate prodrugs of (-)-beta-d-(2R,4R)-dioxolane-thymine: Synthesis, anti-HIV activity and stability studies
Liang, Y, Narayanasamy, J, Schinazi, RF, and Chu, CK
Bioorg Med Chem 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16314108&dopt=abstract
7. 48225 HIV-LS-337; PUBMED-HIV-12/12/2005
Synthesis and anti-HIV activity of bi-functional betulinic acid derivatives
Huang, L, Ho, P, Lee, KH, and Chen, CH
Bioorg Med Chem 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16314103&dopt=abstract
8. 48226 HIV-LS-337; PUBMED-HIV-12/12/2005
The antiviral activity, mechanism of action, clinical significance and resistance of abacavir in the treatment of pediatric AIDS
Melroy, J and Nair, V
Curr Pharm Des 2005. 11(29): 3847-52
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16305515&dopt=abstract
9. 48227 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Methods and compositions for the inhibition of HIV-1 replication in hum an cells using inhibitors of p21/CDKN1A activity or gene expression, and anti-AIDS uses
Wahl, Sharon M, Vazquez-Maldonado, Nancy, and Greenwell-Wild, Teresa
PATENT: WO 2005046732 ISSUE DATE: 20050526
APPLICATION: 2004 PP: 98 pp.
ASSIGNEE: (The United Sates of America as Represented by the Secretary of Health and Human Services, NIH USA
10. 48228 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Novel 4-oxoquinoline compound and use thereof as hiv integrase inhibitor
Satoh, Motohide, Matsuda, Takashi, Okuda, Satoshi, Kawakami, Hiroshi, Aramaki, Hisateru, Shinkai, Hisashi, Matsuzaki, Yuji, Watanabe, Wataru, Yamataka, Kazunobu, Kiyonari, Shinichi, Wamaki, Shuichi, Takahashi, Mitsuru, Yamada, Naohito, and Nagao, Akemi
PATENT: WO 2005113509 ISSUE DATE: 20051201
APPLICATION: 2005
ASSIGNEE: (Japan Tobacco Inc., Japan
11. 48229 HIV-LS-337; SCIFINDER-HIV-12/5/2005
HIV integrase inhibitors
Wai, John S, Vacca, Joseph P, Zhuang, Linghang, Kim, Boyoung, Lyle, Terry A, Wiscount, Catherine M, Egbertson, Melissa S, Neilson, Lou Anne, Embrey, Mark, Fisher, Thorsten E, and Staas, Donnette D
PATENT: WO 2005110415 ISSUE DATE: 20051124
APPLICATION: 2005 PP: 76 pp.
ASSIGNEE: (Merck & Co., Inc. USA
12. 48230 HIV-LS-337; PUBMED-HIV-12/12/2005
Intermolecular interactions in the crystal structures of potential HIV-1 integrase inhibitors
Majerz-Maniecka, K, Musiol, R, Nitek, W, Oleksyn, BJ, Mouscadet, JF, Bret, ML, and Polanski, J
Bioorg Med Chem Lett 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16289813&dopt=abstract
13. 48231 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Preparation of aminocarbonylphenyl-5H-pyrazolo-benzoxazinyl-phenyl methanone derivs. as HIV replication inhibitors
Tahri, Abdellah, Michiels, Lieve Emma Jan, Van Acker, Koenraad Lodewijk August, and Surleraux, Dominique Louis Nestor Ghislain
PATENT: WO 2005105810 ISSUE DATE: 20051110
APPLICATION: 2005 PP: 46 pp.
ASSIGNEE: (Tibotec Pharmaceuticals Ltd., Ire.
14. 48232 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Use of racemic nor-calanolide A in preparation of anti-HIV medicines
Wang, Lin, Liu, Gang, Tao, Peizhen, Zhang, Xingquan, Zhang, Tian, Huang, Biao, and Zhao, Zhizhong
PATENT: CN 1565442 ISSUE DATE: 20050119
APPLICATION: 2003-11440 PP: 17 pp.
ASSIGNEE: (Institute of Materia Medica, Chinese Academy of Medical Sciences Peop. Rep. China
15. 48233 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Preparation of purine derivatives as antiviral agents
Wang, Xuechao, Liu, Zhongrong, Li, Bogang, Wu, Fengwei, Zhong, Chaobin, He, Min, and Huang, Yu
PATENT: CN 1566118 ISSUE DATE: 20050119
APPLICATION: 2003-4232 PP: 15 pp.
ASSIGNEE: (Chengdu Diao Pharmaceutical Group Co., Ltd. Peop. Rep. China
16. 48234 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Preparation of substituted alkylamides as antiviral agents
Kaplan, Eliahu, Bittner, Shmuel, and Harlev, Eliakim
PATENT: WO 2005092305 ISSUE DATE: 20051006
APPLICATION: 2005 PP: 83 pp.
ASSIGNEE: (New Era Biotech Ltd., Virgin I. Brit.
17. 48235 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Preparation of hydroxynaphthyridinediones as HIV integrase inhibitors
Han, Wei, Egbertson, Melissa, Wai, John S, Zhuang, Linghang, Ruzek, Rowena D, Perlow, Debra S, and Obligado, Vanessa E
PATENT: WO 2005087767 ISSUE DATE: 20050922
APPLICATION: 2005 PP: 83 pp.
ASSIGNEE: (Merck & Co., Inc. USA
18. 48236 HIV-LS-337; SCIFINDER-HIV-12/5/2005
Preparation of N-arylmethyl or N-heterocyclylmethyl-N-(imidazol-2-ymethyl)amines as antagonists of chemokine receptor CXCR4
Saitou, Atsushi, Kikumoto, Shigeyuki, Ono, Masahiro, Matsui, Ryo, Yamamoto, Masashi, Sawa, Tomohiro, Suzuki, Shigeru, and Yanaka, Mikiro
PATENT: WO 2005085209 ISSUE DATE: 20050915
APPLICATION: 2005 PP: 252 pp.
ASSIGNEE: (Kureha Chemical Industry Company, Limited Japan
19. 48237 HIV-LS-337; WOS-HIV-12/4/2005
A short synthetic route to biologically active (+/-)-daurichromenic acid as highly potent anti-HIV agent
Lee, YR and Wang, X
ORGANIC & BIOMOLECULAR CHEMISTRY 2005. 3(21): 3955-3957, 3
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000233241900017
20. 48238 HIV-LS-337; WOS-HIV-12/4/2005
Amino acid derivatives, part 3: New peptide and glycopeptide derivatives conjugated naphthalene. Synthesis, antitumor, anti-HIV, and BVDV evaluation
Al-Masoudi, NA, Al-Masoudi, IA, Ali, IAI, Saeed, B, and La, Colla P
HETEROATOM CHEMISTRY 2005. 16(7): 576-586, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000233369500007
21. 48239 HIV-LS-337; WOS-HIV-12/4/2005
Synthesis of novel 4 'alpha-phenyl and 5 'alpha-methyl branched carbocyclic nucleosides
Oh, CH and Hong, JH
BULLETIN OF THE KOREAN CHEMICAL SOCIETY 2005. 26(10): 1520-1524, 5
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000233211900012
22. 48240 HIV-LS-337; WOS-HIV-12/11/2005
Synthesis, spectroscopic, electrochemical and anti-HIV studies of some mononuclear and dinuclear Fe-III complexes of 3-hydroxy-4 '-benzyloxy flavone containing oxygen, nitrogen and sulphur donors as co-ligands
Mishra, L, Singh, AK, and Maeda, Y
JOURNAL OF THE INDIAN CHEMICAL SOCIETY 2005. 82(10): 879-885, 7
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000233470300003
23. 48241 HIV-LS-337; WOS-HIV-12/11/2005
Analogues of N-terminal truncated synthetic peptide fragments derived from RANTES inhibit HIV-1 infectivity
Ramnarine, EJ, DeViCo, AL, and Vigil-Cruz, SC
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2006. 16(1): 93-95, 3
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000233516200018
24. 48242 HIV-LS-337; WOS-HIV-12/11/2005
The broad anti-viral agent glycyrrhizin directly modulates the fluidity of plasma membrane and HIV-1 envelope
Harada, S
BIOCHEMICAL JOURNAL 2005. 392: 191-199, 9
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000233542800021