ONLINE DATABASE SEARCH - HIV-LS-329-MEMO
1. 47765 HIV-LS-329; PUBMED-HIV-8/23/2005
Novel 8-Substituted Dipyridodiazepinone Inhibitors with a Broad-Spectrum of Activity against HIV-1 Strains Resistant to Non-nucleoside Reverse Transcriptase Inhibitors
O'meara, JA, Yoakim, C, Bonneau, PR, Bos, M, Cordingley, MG, Deziel, R, Doyon, L, Duan, J, Garneau, M, Guse, I, Landry, S, Malenfant, E, Naud, J, Ogilvie, WW, Thavonekham, B, and Simoneau, B
J Med Chem 2005. 48(17): 5580-8
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16107158&dopt=abstract
2. 47766 HIV-LS-329; PUBMED-HIV-8/23/2005
Effect of naturally-occurring gp41 HR1 variations on susceptibility of HIV-1 to fusion inhibitors
Chinnadurai, R, Munch, J, and Kirchhoff, F
AIDS 2005. 19 (13): 1401-5
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16103771&dopt=abstract
3. 47767 HIV-LS-329; SCIFINDER-HIV-8/15/2005
HIV protease inhibitors with potential for once-daily dosing and reduced side effects
DeGoey, David A, Flosi, William J, Grampovnik, David J, Flentge, Charles A, Klein, Larry L, Yeung, Clinton M, Dekhtyar, Tatyana, Colletti, Lynn, Waring, Jeffrey F, Ciurlionis, Rita, Marsh, Kennan C, Schmidt, James M, Swanson, Sue J, Stoll, Vincent, Mamo, Mulugeta, Mo, Hongmei, Kati, Warren M, Molla, Akhteruzzaman, and Kempf, Dale J
Abstracts of Papers, 230th ACS National Meeting, Washington, DC, United States, Aug. 28-Sept. 1, 2005 2005.: MEDI-189
4. 47768 HIV-LS-329; PUBMED-HIV-8/23/2005
A non-natural dinucleotide containing an isomeric L-related deoxynucleoside: dinucleotide inhibitors of anti-HIV integrase activity
Newton, MG, Campana, CF, Chi, GC, Lee, D, Liu, ZJ, Nair, V, Phillips, J, Rose, JP, and Wang, BC
Acta Crystallogr C 2005. 61(Pt 8): 518-20
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16082106&dopt=abstract
5. 47769 HIV-LS-329; PUBMED-HIV-8/23/2005
HIV-1 protease inhibitor induces growth arrest and apoptosis of human prostate cancer LNCaP cells in vitro and in vivo in conjunction with blockade of androgen receptor STAT3 and AKT signaling
Yang, Y, Ikezoe, T, Takeuchi, T, Adachi, Y, Ohtsuki, Y, Takeuchi, S, Koeffler, HP, and Taguchi, H
Cancer Sci 2005. 96(7): 425-33
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=16053514&dopt=abstract
6. 47770 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Antimicrobial activity from medicinal mushrooms
Stamets, Paul
PATENT: WO 2005067955 ISSUE DATE: 20050728
APPLICATION: 2005
ASSIGNEE: (USA)
7. 47771 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Allophenylnorstatine-containing HIV-1 protease inhibitors: design, synthesis and structure-activity relationships for selected P2 ligands
Abdel-Rahman, Hamdy M, El-Koussi, Nawal A, Alkaramany, Gamal S, Youssef, Adel F, and Kiso, Yoshiaki
Bulletin of Pharmaceutical Sciences, Assiut University 2005. 28(1): 95-103
8. 47772 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Preparation of amino acid hydrazide derivatives as HIV protease inhibitors
Randolph, John T, Chen, Hui-ju, Degoey, David A, Flentge, Charles A, Flosi, William J, Grampovnik, David J, Huang, Peggy P, Hutchinson, Douglas K, Kempf, Dale J, Klein, Larry L, and Yeung, Ming C
PATENT: US 20050159469 ISSUE DATE: 20050721
APPLICATION: 2004-10177 PP: 155 pp.
ASSIGNEE: (USA)
9. 47773 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Preparation of non-nucleotide reverse transcriptase inhibitors
Sund, Christian, Roue, Nathalie, Lindstroem, Stefan, Antonov, Dmitry, Sahlberg, Christer, and Jansson, Katarina
PATENT: WO 2005066131 ISSUE DATE: 20050721
APPLICATION: 2004 PP: 118 pp.
ASSIGNEE: (Medivir AB, Swed.
10. 47774 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Preparation of phosphonate analogs of HIV protease inhibitors and methods for identifying anti-HIV therapeutic compounds
Arimilli, Murty N, Becker, Mark M, Birkus, Gabriel, Bryant, Clifford, Chen, James M, Chen, Xiaowu, Cihlar, Tomas, Dastgah, Azar, Eisenberg, Eugene J, Fardis, Maria, Hatada, Marcos, He, Gong-Xin, Jin, Haolun, Kim, Choung U, Lee, William A, Lee, Christopher P, Lin, Kuei-Ying, Liu, Hongtao, Mackman, Richard L, McDermott, Martin J, Mitchell, Michael L, Nelson, Peter H, Pyun, Hyung-Jung, Rowe, Tanisha D, Sparacino, Mark, Swaminathan, Sundaramoorthi, Tario, James D, Wang, Jianying, Williams, Matthew A, Xu, Lianhong, Yang, Zheng-Yu, Yu, Richard H, Zhang, Jiancun, and Zhang, Lijun
PATENT: WO 2005064008 ISSUE DATE: 20050714
APPLICATION: 2004 PP: 1723 pp.
ASSIGNEE: (Gilead Sciences, Inc. USA
11. 47775 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Preparation of amino acid derivatives as HIV protease inhibitors
Degoey, David A, Flentge, Charles A, Flosi, William J, Grampovnik, David J, Kempf, Dale J, Klein, Larry L, Yeung, Ming C, Randolph, John T, Wang, Xiu C, and Yu, Su
PATENT: US 2005148623 ISSUE DATE: 20050707
APPLICATION: 2004-8713 PP: 279 pp.
ASSIGNEE: (USA)
12. 47776 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Virus isolates during acute and chronic human immunodeficiency virus type 1 infection show distinct patterns of sensitivity to entry inhibitors
Rusert, Peter, Kuster, Herbert, Joos, Beda, Misselwitz, Benjamin, Gujer, Cornelia, Leemann, Christine, Fischer, Marek, Stiegler, Gabriela, Katinger, Hermann, Olson, William C, Weber, Rainer, Aceto, Leonardo, Guenthard, Huldrych F, and Trkola, Alexandra
Journal of Virology 2005. 79(13): 8454-8469
13. 47777 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Antiviral protein OVT102 derived from cyanovirin with improved properties and methods therefor
Levine, Howard L and Kerns, William
PATENT: WO 2005058229 ISSUE DATE: 20050630
APPLICATION: 2004 PP: 32 pp.
ASSIGNEE: (Omniviral Therapeutics LLC, USA
14. 47778 HIV-LS-329; SCIFINDER-HIV-8/15/2005
HIV (human immunodeficiency virus) gp41 mimetibodies as improved anti-retroviral agents with longer plasma half-lives, and therapeutic uses thereof
Dillon, Susan B, Del Vecchio, Alfred Michael, Huang, Chichi, O'Neil, Karyn T, and Sarisky, Robert T
PATENT: US 2005136061 ISSUE DATE: 20050623
APPLICATION: 2004-18102 PP: 18 pp.
ASSIGNEE: (USA)
15. 47779 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Carbazole derivatives as integrase inhibitors and anti-retrovirus medicines
Chiba, Tomoko, Yan, Ka, and Sugiura, Yuzuru
PATENT: JP 2005154347 ISSUE DATE: 20050616
APPLICATION: 2003-2643 PP: 16 pp.
ASSIGNEE: (Toyama Chemical Co., Ltd. Japan
16. 47780 HIV-LS-329; WOS-HIV-8/14/2005
Nonnucleoside HIV-1 reverse transcriptase inhibitors, part 4. Synthesis and anti-HIV activity of N-1-beta-carbonyl-6-naphthylmethyl analogues of HEPT
He, YP, Kuang, YY, Chen, F, Wang, SX, Ji, L, De, Clercq E, Balzarini, J, and Pannecouque, C
MONATSHEFTE FUR CHEMIE 2005. 136(7): 1233-1245, 13
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000230819000010
17. 47781 HIV-LS-329; WOS-HIV-8/14/2005
Synthesis of N-1-(indanyloxymethyl) and N-1-(4-hydroxybut-2-enyloxymethyl) analogues of the HIV drugs Emivirine and GCA-186
El-Brollosy, NR, Nielsen, C, and Pedersen, EB
MONATSHEFTE FUR CHEMIE 2005. 136(7): 1247-1254, 8
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000230819000011
18. 47782 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Antiviral compositions for treatment of HIV infection
Wood, Allen Wayne, Currie, Robin, Mehta, Samir Chimanlal, Goodson, Gary Wayne, and Wells, Mickey Lee
PATENT: US 2005113394 ISSUE DATE: 20050526
APPLICATION: 2004-14360 PP: 6 pp.
ASSIGNEE: (USA)
19. 47783 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Anti-HIV Activity of (-)-(2R,4R)-1- (2-Hydroxymethyl-1,3-dioxolan-4-yl)thymine against Drug-Resistant HIV-1 Mutants and Studies of Its Molecular Mechanism
Chu, Chung K, Yadav, Vikas, Chong, Youhoon H, and Schinazi, Raymond F
Journal of Medicinal Chemistry 2005. 48(12): 3949-3952
20. 47784 HIV-LS-329; SCIFINDER-HIV-8/15/2005
Structure-Based Design: Synthesis and Biological Evaluation of a Series of Novel Cycloamide-Derived HIV-1 Protease Inhibitors
Ghosh, Arun K, Swanson, Lisa M, Cho, Hanna, Leshchenko, Sofiya, Hussain, Khaja Azhar, Kay, Stephanie, Walters, DEric, Koh, Yasuhiro, and Mitsuya, Hiroaki
Journal of Medicinal Chemistry 2005. 48(10): 3576-3585
21. 47785 HIV-LS-329; WOS-HIV-8/21/2005
Combinatorial selection, inhibition, and antiviral activity of DNA thioaptamers targeting the RNase H domain of HIV-1 reverse transcriptase
Somasunderam, A, Ferguson, MR, Rojo, DR, Thiviyanathan, V, Li, X, O'Brien, WA, and Gorenstein, DG
BIOCHEMISTRY 2005. 44(30): 10388-10395, 8
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000230879900044