ONLINE DATABASE SEARCH - HIV-LS-319-MEMO
1. 45079 HIV-LS-319; PUBMED-HIV-4/5/2005
Synthesis of 2',3'-Dideoxynucleoside 5'-alpha-P-Borano-beta,gamma-(difluoromethylene)triphosphates and Their Inhibition of HIV-1 Reverse Transcriptase
Boyle, NA, Rajwanshi, VK, Prhavc, M, Wang, G, Fagan, P, Chen, F, Ewing, GJ, Brooks, JL, Hurd, T, Leeds, JM, Bruice, TW, and Cook, PD
J Med Chem 2005. 48(7): 2695-2700
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15801860&dopt=abstract
2. 45080 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Selective Small Molecules Blocking HIV-1 Tat and Coactivator PCAF Association
Zeng, Lei, Li, Jiaming, Muller, Michaela, Yan, Sherry, Mujtaba, Shiraz, Pan, Chongfeng, Wang, Zhiyong, and Zhou, Ming-Ming
Journal of the American Chemical Society 2005. 127(8): 2376-2377
3. 45081 HIV-LS-319; PUBMED-HIV-4/5/2005
Simple and Simultaneous Determination of the HIV-Protease Inhibitors Amprenavir, Atazanavir, Indinavir, Lopinavir, Nelfinavir, Ritonavir and Saquinavir Plus M8 Nelfinavir Metabolite and the Nonnucleoside Reverse Transcriptase Inhibitors Efavirenz and Nevirapine in Human Plasma by Reversed-Phase Liquid Chromatography
Poirier, JM, Robidou, P, and Jaillon, P
Ther Drug Monit 2005. 27(2): 186-192
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15795650&dopt=abstract
4. 45082 HIV-LS-319; PUBMED-HIV-4/5/2005
Peptides derived from the reverse transcriptase of human immunodeficiency virus type 1 as novel inhibitors of the viral integrase
Oz-Gleenberg, I, Avidan, O, Goldgur, Y, Herschhorn, A, and Hizi, A
J Biol Chem 2005.
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15790559&dopt=abstract
5. 45083 HIV-LS-319; PUBMED-HIV-4/5/2005
The antimicrobial peptide dermaseptin S4 inhibits HIV-1 infectivity in vitro
Lorin, C, Saidi, H, Belaid, A, Zairi, A, Baleux, F, Hocini, H, Belec, L, Hani, K, and Tangy, F
Virology 2005. 334(2): 264-275
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15780876&dopt=abstract
6. 45084 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Synthesis and Evaluation of Double-Prodrugs against HIV. Conjugation of D4T with 6-Benzyl-1-(ethoxymethyl)-5-isopropyluracil (MKC-442, Emivirine)-Type Reverse Transcriptase Inhibitors via the SATE Prodrug Approach
Petersen, Lene, Jorgensen, Per T, Nielsen, Claus, Hansen, Thomas H, Nielsen, John, and Pedersen, Erik B
Journal of Medicinal Chemistry 2005. 48(4): 1211-1220
7. 45085 HIV-LS-319; PUBMED-HIV-4/5/2005
4-Benzyl and 4-benzoyl-3-dimethylaminopyridin-2(1H)-ones: in vitro evaluation of new C-3-amino-substituted and C-5,6-alkyl-substituted analogues against clinically important HIV Mutant Strains
Benjahad, A, Croisy, M, Monneret, C, Bisagni, E, Mabire, D, Coupa, S, Poncelet, A, Csoka, I, Guillemont, J, Meyer, C, Andries, K, Pauwels, R, de, Bethune MP, Himmel, DM, Das, K, Arnold, E, Nguyen, CH, and Grierson, DS
J Med Chem 2005. 48(6): 1948-1964
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15771439&dopt=abstract
8. 45086 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Identification of authentic inhibitors of HIV-1 integration
Witvrouw, M, Fikkert, V, Vercammen, J, Van Maele, B, Engelborghs, Y, and Debyser, Z
Current Medicinal Chemistry: Anti-Infective Agents 2005. 4(2): 153-165
9. 45087 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Hiv protease inhibitors, compositions containing the same and their pharmaceutical uses
Alegria, Larry Andrew, Dress, Klaus Ruprecht, Huang, Buwen, Kumpf, Robert Arnold, Lewis, Kathleen Kingsley, Matthews, Jean Joo, Sakata, Sylvie Kim, and Wallace, Michael Brennan
PATENT: WO 2005026114 ISSUE DATE: 20050324
APPLICATION: 2004
ASSIGNEE: (Pfizer Inc., USA
10. 45088 HIV-LS-319; SCIFINDER-HIV-3/29/2005
The Novel L- and D-Amino Acid Derivatives of Hydroxyurea and Hydantoins: Synthesis, X-ray Crystal Structure Study, and Cytostatic and Antiviral Activity Evaluations
Opacic, Ninoslav, Barbaric, Monika, Zorc, Branka, Cetina, Mario, Nagl, Ante, Frkovic, Danijel, Kralj, Marijeta, Pavelic, Kresimir, Balzarini, Jan, Andrei, Graciela, Snoeck, Robert, De Clercq, Erik, Raic-Malic, Silvana, and Mintas, Mladen
Journal of Medicinal Chemistry 2005. 48(2): 475-482
11. 45089 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Synthesis and antiviral activity of novel 4',5'-branched pyrimidine nucleosides
Kim, Aihong, Kooh, Dae-Ho, Ko, Ok Hyun, and Hong, Joon Hee
Yakhak Hoechi 2005. 49(1): 20-24
12. 45090 HIV-LS-319; PUBMED-HIV-4/5/2005
Nuclear translocation as a novel target for anti-HIV drugs
Haffar, O and Bukrinsky, M
Expert Rev Anti Infect Ther 2005. 3(1): 41-50
HYPERLINK:
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=15757456&dopt=abstract
13. 45091 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Compositions and methods for use of antiviral drugs in the treatment of retroviral diseases resistant to nucleoside reverse transcriptase inhibitors
Parniak, Michael, Mellors, John W, Oldfield, Eric, Tovian, Zev, and Chan, Julian Mun Weng
PATENT: WO 2005023270 ISSUE DATE: 20050317
APPLICATION: 2004 PP: 50 pp.
ASSIGNEE: (University of Pittsburgh-of the Commonwealth System of Higher Education, USA and University of Illinois)
14. 45092 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Combinations of pyrimidine-containing nonnucleoside reverse transcriptase inhibitor (NNRTI) TMC278 with reverse transcriptase inhibitors for the treatment of HIV infection
Stoffels, Paul
PATENT: WO 2005021001 ISSUE DATE: 20050310
APPLICATION: 2004 PP: 34 pp.
ASSIGNEE: (Tibotec Pharmaceuticals Ltd., Ire.
15. 45093 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Structure activity relationship of disulfone-containing HIV-1 integrase inhibitors
Meadows, DChristopher, Gervay-Hague, Jacquelyn, Matthews, Timothy B, and North, Thomas W
229th ACS National Meeting 2005. 229: MEDI-338
16. 45094 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Discovery of the piperidine-4-carboxamide derivative TAK-220, a highly potent CCR5 antagonist anti-HIV-1 agent
Imamura, Shinichi, Ichikawa, Takashi, Nishikawa, Youichi, Hashiguchi, Shohei, Kanzaki, Naoyuki, Takashima, Katsunori, Niwa, Shinichi, Yamamoto, Yoshio, Baba, Masanori, and Sugihara, Yoshihiro
229th ACS National Meeting 2005. 229: MEDI-090
17. 45095 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Structural and Functional Modeling of Human Lysozyme Reveals a Unique Nonapeptide, HL9, with Anti-HIV Activity
Lee-Huang, Sylvia, Maiorov, Vladimir, Huang, Philip L, Ng, Angela, Lee, Hee Chul, Chang, Young-Tae, Kallenbach, Neville, Huang, Paul L, and Chen, Hao-Chia
Biochemistry 2005. 44(12): 4648-4655
18. 45096 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Novel HIV integrase inhibitors and HIV therapy based on drug combinations including integrase inhibitors
Robinson, WEdward, King, Peter J, and Reinecke, Manfred G
PATENT: US 20050049242 ISSUE DATE: 20050303
APPLICATION: 2003-17364 PP: 32 pp., Cont. of U.S. Ser. No. 647,270, abandoned.
ASSIGNEE: (USA)
19. 45097 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Preparation of pyrido[1,2-a]pyrazine-1,8-dione derivatives as HIV integrase inhibitors
Miyazaki, Susumu, Katoh, Susumu, Adachi, Kaoru, Isoshima, Hirotaka, Kobayashi, Satoru, Matsuzaki, Yuji, Watanabe, Wataru, Yamataka, Kazunobu, Kiyonari, Shinichi, and Wamaki, Shuichi
PATENT: WO 2005016927 ISSUE DATE: 20050224
APPLICATION: 2004 PP: 355 pp.
ASSIGNEE: (Japan Tobacco Inc., Japan
20. 45098 HIV-LS-319; SCIFINDER-HIV-3/29/2005
Topological models for the prediction of anti-HIV activity of dihydro (alkylthio) (naphthylmethyl) oxopyrimidines
Lather, Viney and Madan, AK
Bioorganic & Medicinal Chemistry 2005. 13(5): 1599-1604
21. 45099 HIV-LS-319; WOS-HIV-3/27/2005
Exploring the stereochemical requirements for protease inhibition by ureidopeptides
Barth, BS, Myers, AC, and Lipton, MA
JOURNAL OF PEPTIDE RESEARCH 2005. 65(3): 352-354, 3
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227499400005
22. 45100 HIV-LS-319; WOS-HIV-3/27/2005
HIV-1 Vif can directly inhibit apolipoprotein B mRNA-editing enzyme catalytic polypeptide-like 3G-mediated cytidine deamination by using a single amino acid interaction and without protein degradation
Santa-Marta, M, da, Silva FA, Fonseca, AM, and Goncalves, J
JOURNAL OF BIOLOGICAL CHEMISTRY 2005. 280(10): 8765-8775, 11
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227453100019
23. 45101 HIV-LS-319; WOS-HIV-3/27/2005
Racemic and enantioselective synthesis of enol-lactone and their biological activity as potent HIV-1 protease inhibitors
Ibrahimi, S, Sauve, G, Yelle, J, and Essassi, E
COMPTES RENDUS CHIMIE 2005. 8(1): 75-83, 9
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227238000010
24. 45102 HIV-LS-319; WOS-HIV-3/27/2005
Synthesis of racemic 9-(6-and 2,6-substituted 9H-purin-9-yl)-5-oxatricyclo[4.2.1.0(3,7)]non ne-3-methanols, novel conformationally locked carbocyclic nucleosides
Hrebabecky, H, Masojidkova, M, and Holy, A
COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS 2005. 70(1): 103-123, 21
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227529600009
25. 45103 HIV-LS-319; WOS-HIV-3/27/2005
A novel synthetic chemokine containing D-amino acids that binds to the CXCR4 receptor and inhibits HIV-1 infection
Huang, ZW, Liu, DX, Madani, N, Kumar, S, Choi, WT, Cao, R, Li, Y, Gao, YG, Dong, CZ, Wang, J, An, J, and Sodroski, JG
BLOOD 2004. 104(11): 174A-1
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000225127500606
26. 45104 HIV-LS-319; WOS-HIV-4/3/2005
Plant based HIV-1 vaccine candidate: Tat protein produced in spinach
Karasev, AV, Foulke, S, Wellens, C, Rich, A, Shon, KJ, Zwierzynski, I, Hone, D, Koprowski, H, and Reitz, M
VACCINE 2005. 23(15): 1875-1880, 6
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227769600024
27. 45105 HIV-LS-319; WOS-HIV-4/3/2005
HIV-1 replication inhibitors of the styrylquinoline class: introduction of an additional carboxyl group at the C-5 position of the quinoline
Zouhiri, F, Danet, M, Benard, C, Normand-Bayle, M, Mouscadet, JF, Leh, H, Thomas, CM, Mbemba, G, d'Angelo, J, and Desmaele, D
TETRAHEDRON LETTERS 2005. 46(13): 2201-2205, 5
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000227754000006