ONLINE DATABASE SEARCH -
HIV-LS-383-MEMO
1.
61638 HIV-LS-383;
WOS-HIV-9/7/2007
Synthesis of 2-Benzothienyl Carbonyl 4-Arylpiperazines as Novel
Delavirdine Analogs
Pessoa-Mahana, H. et al.
Synthetic Communications 2007. 37(7-9): 1227-1235
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000247620500020
2.
61639 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
CCR5 antagonists useful for treating HIV
Ramanathan, Ragulan, Miller, Michael W, Chowdhury, Swapan K, Alton, Kevin
B, Grotz, Diane, Rindgen, Diane, and Tendolkar, Amol
PATENT: US 2007203149 ISSUE DATE: 20070830
APPLICATION: 2007-22529 PP:
17pp.
ASSIGNEE: (Schering
Corporation, USA
View Data on the NIAID Therapeutics Website
HYPERLINK:
3.
61640 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Pyridin-2(1H)-ones: a promising class of HIV-1 non-nucleoside reverse
transcriptase inhibitors
Medina-Franco, Jose Luis, Martinez-Mayorga, Karina, Juarez-Gordiano,
Cecilia, and Castillo, Rafael
ChemMedChem 2007.
2(8): 1141-1147
View Data on the NIAID Therapeutics Website
HYPERLINK:
4.
61641 HIV-LS-383;
WOS-HIV-9/7/2007
Human Polycomb Group Eed Protein Negatively Affects Hiv-1 Assembly and
Release
Rakotobe, D. et al.
Retrovirology 2007.
4
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000247632900001
5.
61642 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
pyrrolo[3,4-c]pyrrole derivatives as heterocyclic antiviral compounds and
CCR5 receptor antagonists and their preparation, pharmaceutical compositions and
use in the treatment of HIV infection, AIDS and ARC
Lemoine, Rcmy, Melville, Chris Richard, Padilla, Fernando, Rotstein,
David Mark, and Wanner, Jutta
PATENT: US
2007191406 ISSUE DATE: 20070816
APPLICATION: 2007-51368 PP:
45pp.
ASSIGNEE: (Roche Palo Alto
LLC, USA
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HYPERLINK:
6.
61643 HIV-LS-383;
WOS-HIV-9/7/2007
Ccr5 Small-Molecule Antagonists and Monoclonal Antibodies Exert Potent
Synergistic Antiviral Effects by Cobinding to the Receptor
Ji, C. et al.
Molecular Pharmacology 2007.
72(1): 18-28
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000247477600003
7.
61644 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Use of
6-(3-chloro-2-fluorobenzyl)-1-[(2S)-1-hydroxy-3-methylbutan-2-yl]-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic
acid or salt thereof for treating retrovirus infection
Matsuzaki, Yuji, Kano, Mitsuki, and Ikeda, Satoru
PATENT: WO
2007089030 ISSUE DATE: 20070809
APPLICATION: 2007 PP:
89pp.
ASSIGNEE: (Japan Tobacco
Inc., Japan
View Data on the NIAID Therapeutics Website
HYPERLINK:
8.
61645 HIV-LS-383;
WOS-HIV-9/7/2007
Rational Optimization of the Binding Affinity of Cd4 Targeting
Peptidomimetics With Potential Anti Hiv Activity
Neffe, A. et al.
Journal of Medicinal Chemistry 2007. 50(15): 3482-3488
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000248121300012
9.
61646 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Preparation of imidazo[1,2-a]pyridine compds. useful in the treatment of
HIV infection and other chemokine receptor-mediated diseases
Gudmundsson, Kristjan, Boggs, Sharon Davis, Miller, John Franklin, and
Svolto, Angilique Christina
PATENT: WO
2007087549 ISSUE DATE: 20070802
APPLICATION: 2007 PP:
148pp.
ASSIGNEE: (Smithkline
Beecham Corporation, USA
View Data on the NIAID Therapeutics Website
HYPERLINK:
10.
61647 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Imidazo[1,2-a]pyridine-3-carboxamides as anti-HIV agents and their
preparation, pharmaceutical compositions and their use in monotherapy and in
combination therapy of diseases
Gudmundsson, Kristjan and Turner, Elizabeth
Madalena
PATENT: WO 2007087548 ISSUE DATE: 20070802
APPLICATION: 2007 PP:
104pp.
ASSIGNEE: (Smithkline
Beecham Corporation, USA and Svolto, Angilique
Christina
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HYPERLINK:
11.
61648 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Synthesis of 8-halogenated adenosine compounds as antiviral
agents
Chang, Junbiao, Cheng, Senxiang, Wang, Limin, Hao, Jia, Wang, Qiang, and
Guo, Xiaohe
PATENT: CN
101003550 ISSUE DATE:
20070725
APPLICATION: 1016-30 PP:
14pp.
ASSIGNEE: (Henan Center of
Analysis and Test, Peop. Rep. China
View Data on the NIAID Therapeutics Website
HYPERLINK:
12.
61649 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Design and cellular kinetics of dansyl-labeled CADA derivatives with
anti-HIV and CD4 receptor down-modulating activity
Vermeire, Kurt, Lisco, Andrea, Grivel, Jean-Charles, Scarbrough, Emily,
Dey, Kaka, Duffy, Noah, Margolis, Leonid, Bell, Thomas W, and Schols,
Dominique
Biochem. Pharmacol. 2007.
74(4): 566-578
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HYPERLINK:
13.
61650 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Hologram quantitative structure-activity relationships for a class of
inhibitors of HIV-1 protease
Ferreira, Leonardo G, Leitao, Andrei, Montanari, Carlos A, and
Andricopulo, Adriano D
Lett. Drug Des. Discovery 2007. 4(5): 356-364
View Data on the NIAID Therapeutics Website
HYPERLINK:
14.
61651 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
A novel bis-tetrahydrofuranylurethane-containing nonpeptidic protease
inhibitor (PI), GRL-98065, is potent against multiple-PI-resistant human
immunodeficiency virus in vitro
Amano, Masayuki, Koh, Yasuhiro, Das, Debananda, Li, Jianfeng, Leschenko,
Sofiya, Wang, Yuan-Fang, Boross, Peter I, Weber, Irene T, Ghosh, Arun K, and
Mitsuya, Hiroaki
Antimicrob. Agents Chemother. 2007. 51(6): 2143-2155
View Data on the NIAID Therapeutics Website
HYPERLINK:
15.
61652 HIV-LS-383;
SCIFINDER-HIV-9/10/2007
Synthesis and anti-HIV-1 activity of new MKC-442 analogues with an
alkynyl-substituted 6-benzyl group
Aly, Youssef L, Pedersen, Erik B, La Colla, Paolo, and Loddo,
Roberta
Arch. Pharm. (Weinheim, Ger.) 2007. 340(5): 225-235
View Data on the NIAID Therapeutics Website
HYPERLINK:
16.
61653 HIV-LS-383;
WOS-HIV-9/7/2007
Pharmacokinetics of the Anti-Human Immunodeficiency Virus Agent
1-(Beta-D-Dioxolane)Thymine in Rhesus Monkeys
Asif, G. et al.
Antimicrobial Agents and Chemotherapy 2007. 51(7): 2424-2429
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000247665800019
17.
61654 HIV-LS-383;
WOS-HIV-9/14/2007
Novel Synthesis and Anti-Hiv-1 Activity of
2-Arylthio-6-Benzyl-2,3-Dihydro-1h-Pyrimidin-4-Ones (Aryl
S-Dabos)
Aly, Y. et al.
Synthesis-Stuttgart 2007.(13): 1955-1960
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000248184200008
18.
61655 HIV-LS-383;
WOS-HIV-9/14/2007
Nuclear Factor 90(Nf90) Targeted to Tar Rna Inhibits Transcriptional
Activation of Hiv-I
Agbottah, E. et al.
Retrovirology 2007.
4
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000248016200002
19.
61656 HIV-LS-383;
WOS-HIV-9/14/2007
Qsar Analysis of Caffeoyl Naphthalene Sulfonamide Derivatives as Hiv-1
Integrase Inhibitors
Sahu, K. et al.
Medicinal Chemistry Research 2007. 15(7-8): 418-430
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000248743400003
20.
61657 HIV-LS-383;
WOS-HIV-9/14/2007
All-Trans Retinoic Acid Attacks Reverse Transcriptase Resulting in
Inhibition of Hiv-1 Replication
Maeda, Y. et al.
Hematology 2007.
12(3): 263-266
View Data on the NIAID Therapeutics Website
HYPERLINK:
http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000248115000013
21.
61658 HIV-LS-383;
PUBMED-HIV-9/17/2007
Discovery and Synthesis of HIV Integrase Inhibitors: Development of
Potent and Orally Bioavailable N-Methyl Pyrimidones
Gardelli, C, Nizi, E, Muraglia, E, Crescenzi, B, Ferrara, M, Orvieto, F,
Pace, P, Pescatore, G, Poma, M, Ferreira, MD, Scarpelli, R, Homnick, CF,
Ikemoto, N, Alfieri, A, Verdirame, M, Bonelli, F, Paz, OG, Taliani, M,
Monteagudo, E, Pesci, S, Laufer, R, Felock, P, Stillmock, KA, Hazuda, D, Rowley,
M, and Summa, V
J Med Chem 2007.
View Data on the NIAID Therapeutics Website
HYPERLINK:
22.
61659 HIV-LS-383;
PUBMED-HIV-9/17/2007
Inhibition of Human Immunodeficiency Virus Type-1 Concerted Integration
by Strand Transfer Inhibitors Which Recognize a Transient Structural
Intermediate
Pandey, KK, Bera, S, Zahm, J, Vora, A, Stillmock, K, Hazuda, D, and
Grandgenett, DP
J Virol 2007.
View Data on the NIAID Therapeutics Website
HYPERLINK:
23.
61660 HIV-LS-383;
PUBMED-HIV-9/17/2007
Identification of potential HIV-1 targets of minocycline
Jenwitheesuk, E and Samudrala, R
Bioinformatics
2007.
View Data on the NIAID Therapeutics Website
HYPERLINK:
24.
61661 HIV-LS-383;
PUBMED-HIV-9/17/2007
Indolyl Aryl Sulfones as HIV-1 Non-Nucleoside Reverse Transcriptase
Inhibitors: Role of Two Halogen Atoms at the Indole Ring in Developing New
Analogues with Improved Antiviral Activity
Regina, GL, Coluccia, A, Piscitelli, F, Bergamini, A, Sinistro, A,
Cavazza, A, Maga, G, Samuele, A, Zanoli, S, Novellino, E, Artico, M, and
Silvestri, R
J Med Chem 2007.
View Data on the NIAID Therapeutics Website
HYPERLINK:
25. 61662
HIV-LS-383;
PUBMED-HIV-9/17/2007
Synthesis and Biological Evaluation of Alkenyldiarylmethane HIV-1
Non-Nucleoside Reverse
Transcriptase Inhibitors That Possess Increased Hydrolytic
Stability
Cullen, MD, Deng, BL, Hartman, TL, Watson, KM, Buckheit, RW Jr,
Pannecouque, C, Clercq, ED, and Cushman, M
J Med Chem 2007.
HYPERLINK:
26.
61663 HIV-LS-383;
PUBMED-HIV-9/17/2007
Fluorescence correlation spectroscopy at single molecule level on the
Tat-TAR complex and its inhibitors
Nandi, CK, Parui, PP,
Brutschy, B, Scheffer, U, and Gobel, M
Biopolymers 2007.
View Data on the NIAID Therapeutics Website
HYPERLINK:
27.
61664 HIV-LS-383;
PUBMED-HIV-9/17/2007
Intracellular Metabolism and Persistence of the Anti-Human
Immunodeficiency Virus Activity of 2', 3'-Didehydro-3'-Deoxy-4'-
Ethynylthymidine, A Novel Thymidine Analog
Paintsil, E, Dutschman, GE, Hu, R, Grill, SP, Lam, W, Baba, M, Tanaka, H,
and Cheng, YC
Antimicrob Agents Chemother 2007.