ONLINE DATABASE SEARCH - HIV-LS-375-MEMO

1. 60898 HIV-LS-375; SCIFINDER-HIV-5/21/2007

Tmaz as an antiviral agent and use thereof

Lelas, Tihomir

PATENT: WO 2007054085 ISSUE DATE: 20070518

APPLICATION: 2006

ASSIGNEE: (Ljubicic, Mijo Germany and Ivkovic, Slavko

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2. 60899 HIV-LS-375; SCIFINDER-HIV-5/21/2007

Agaritine and its derivatives are potential inhibitors against HIV proteases

Gao, Wei-Na, Wei, Dong-Qing, Li, Yun, Gao, Hui, Xu, Wei-Ren, Li, Ai-Xiu, and Chou, Kuo-Chen

Med. Chem. 2007. 3(3): 221-226

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3. 60900 HIV-LS-375; PUBMED-HIV-5/29/2007

Human immunodeficiency virus type 1 Vif inhibits packaging and antiviral activity of a degradation-resistant APOBEC3G variant

Opi, S, Kao, S, Goila-Gaur, R, Khan, MA, Miyagi, E, Takeuchi, H, and Strebel, K

J Virol 2007.

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17522211&dopt=abstract

4. 60901 HIV-LS-375; PUBMED-HIV-5/29/2007

An alternative strategy for inhibiting multidrug-resistant mutants of the dimeric HIV-1 protease by targeting the subunit interface

Bannwarth, L and Reboud-Ravaux, M

Biochem Soc Trans 2007. 35(Pt 3): 551-4

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17511649&dopt=abstract

5. 60902 HIV-LS-375; PUBMED-HIV-5/29/2007

A Naturally Occurring Splice Variant of CXCL12/Stromal Cell-Derived Factor 1 is a potent HIV-1 Inhibitor with Weak Chemotaxis and Cell Survival Activities

Altenburg, JD, Broxmeyer, HE, Jin, Q, Cooper, S, Basu, S, and Alkhatib, G

J Virol 2007.

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17507482&dopt=abstract

6. 60903 HIV-LS-375; SCIFINDER-HIV-5/21/2007

Small molecule inhibitors of HIV-1 capsid assembly

Prevelige, Peter Jr

PATENT: WO 2007048042 ISSUE DATE: 20070426

APPLICATION: 2006 PP: 69pp.

ASSIGNEE: (University of Alabama at Birmingham, USA

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7. 60904 HIV-LS-375; SCIFINDER-HIV-5/21/2007

Use of bivalent or polyvalent trisaccharides as fusion inhibitors in all HIV types, subtypes, groups, strains, and circulating recombinant forms, as well as for the treatment of other viral infections and cancer

Farquharson, Mercedes

PATENT: US 2007093452 ISSUE DATE: 20070426

APPLICATION: 2005-57377 PP: 4pp.

ASSIGNEE: (USA)

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8. 60905 HIV-LS-375; PUBMED-HIV-5/29/2007

QSAR Study on Pyridinone Derivatives as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor: A Mixed Approach

Vasanthanathan, P, Lakshmi, M, and Rao, AR

Med Chem 2007. 3(3): 227-32

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17504193&dopt=abstract

9. 60906 HIV-LS-375; SCIFINDER-HIV-5/21/2007

N-Phenyl-phenylacetamide derivatives as non-nucleoside reverse transcriptase inhibitors, their preparation, pharmaceutical compositions, and use in therapy

Mirzadegan, Taraneh and Silva, Tania

PATENT: US 2007088053 ISSUE DATE: 20070419

APPLICATION: 2006-59058 PP: 27pp.

ASSIGNEE: (Roche Palo Alto LLC, USA

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10. 60907 HIV-LS-375; SCIFINDER-HIV-5/21/2007

N-Phenyl-phenylacetamide derivatives as non-nucleoside reverse transcriptase inhibitors, their preparation, pharmaceutical compositions, and use in therapy

Silva, Tania and Sweeney, Zachary Kevin

PATENT: US 2007088015 ISSUE DATE: 20070419

APPLICATION: 2006-59057 PP: 32pp.

ASSIGNEE: (Roche Palo Alto LLC, USA

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11. 60908 HIV-LS-375; PUBMED-HIV-5/29/2007

A phase I/IIa study with succinylated human serum albumin (Suc-HSA), a candidate HIV-1 fusion inhibitor

Vermeulen, JN, Meijer, DK, Over, J, Lange, J, Proost, JH, Bakker, HI, Beljaars, L, Wit, FW, and Prins, JM

Antivir Ther 2007. 12(2): 273-8

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17503670&dopt=abstract

12. 60909 HIV-LS-375; SCIFINDER-HIV-5/21/2007

Preparation of pyrimidine and pyrimidinone derivatives and their use for the treatment of HIV infections

Botta, Maurizio, Corelli, Federico, Petricci, Elena, Radi, Marco, Maga, Giovanni, Este'a, Jose, and Mai, Antonello

PATENT: WO 2007043094 ISSUE DATE: 20070419

APPLICATION: 2006 PP: 53pp.

ASSIGNEE: (Universita degli Studi di Siena, Italy

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13. 60910 HIV-LS-375; PUBMED-HIV-5/29/2007

Antiretroviral drug resistance, HIV-1 tropism, and HIV-1 subtype among men who have sex with men with recent HIV-1 infection

Eshleman, SH, Husnik, M, Hudelson, S, Donnell, D, Huang, Y, Huang, W, Hart, S, Jackson, B, Coates, T, Chesney, M, and Koblin, B

AIDS 2007. 21 (9): 1165-1174

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17502727&dopt=abstract

14. 60911 HIV-LS-375; SCIFINDER-HIV-5/21/2007

Preparation of heterocyclic Non-nucleoside reverse transcriptase inhibitors

Saito, Yoshihito David, Smith, Mark, and Sweeney, Zachary Kevin

PATENT: US 2007078128 ISSUE DATE: 20070405

APPLICATION: 54 PP: 31pp.

ASSIGNEE: (USA)

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15. 60912 HIV-LS-375; PUBMED-HIV-5/29/2007

Structure-Activity Relationships of Synthetic Coumarins as HIV-1 Inhibitors

Kostova, I, Raleva, S, Genova, P, and Argirova, R

Bioinorg Chem Appl 2006.: 68274

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17497014&dopt=abstract

16. 60913 HIV-LS-375; PUBMED-HIV-5/29/2007

Evaluation of the substrate envelope hypothesis for inhibitors of HIV-1 protease

Chellappan, S, Kairys, V, Fernandes, MX, Schiffer, C, and Gilson, MK

Proteins 2007.

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17474129&dopt=abstract

17. 60914 HIV-LS-375; PUBMED-HIV-5/29/2007

Improved oral bioavailability of anti-HIV agent N'-[2-(2-thiophene)ethyl]-N'-[2-(5-bromopyridyl)]-thiourea (HI-443) in a novel lipophilic formulation

Uckun, FM, Erbeck, D, Tibbles, H, Qazi, S, and Venkatachalam, TK

Arzneimittelforschung 2007. 57(3): 164-70

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http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17469651&dopt=abstract

18. 60915 HIV-LS-375; WOS-HIV-5/18/2007

Synthesis and anti-HIV activity of 4-chloro-2-mercapto-N-(1,4,5,6-tetrahydro-1,2,4-triazin-3-yl)benzenesulf onamide derivatives

Pomarnacka, E

POLISH JOURNAL OF CHEMISTRY 2007. 81(3): 345-352

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http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000245413300005

19. 60916 HIV-LS-375; WOS-HIV-5/18/2007

Design and synthesis of BACE1 inhibitors containing a novel norstatine derivative (2R,3R)-3-amino-2-hydroxy-4(phenylthio)butyric acid

Ziora, Z, Kasai, S, Hidaka, K, Nagamine, A, Kimura, T, Hayashi, Y, and Kiso, Y

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 2007. 17(6): 1629-1633

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http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000245492400029

20. 60917 HIV-LS-375; WOS-HIV-5/18/2007

Novel in vivo model for the study of human immunodeficiency virus type 1 transcription inhibitors: Evaluation of new 6-desfluoroquinolone derivatives

Stevens, M, Pollicita, M, Pannecouque, C, Verbeken, E, Tabarrini, O, Cecchetti, V, Aquaro, S, Perno, CF, Fravolini, A, De Clercq, E, Schols, D, and Balzarini, J

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY 2007. 51(4): 1407-1413

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http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000245416500040

21. 60918 HIV-LS-375; WOS-HIV-5/25/2007

Resistance of HIV-1 to the broadly HIV-1-neutralizing, anti-carbohydrate antibody 2G12

Huskens, D, Van Laethem, K, Vermeire, K, Balzarini, J, and Schols, D

VIROLOGY 2007. 360(2): 294-304

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http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000245566100006

22. 60919 HIV-LS-375; WOS-HIV-5/25/2007

Anti-HIV activity of a cardiac glycoside isolated from Elaeodendron croceum

Prinsloo, G, Meyer, JJM, and Hussein, AA