ONLINE DATABASE SEARCH - HIV-LS-373-MEMO

 

1.     60729   HIV-LS-373; SCIFINDER-HIV-4/23/2007

          Piperazine amidines as antiviral agents

          Wang, Tao, Kadow, John F, Meanwell, Nicholas A, Zhang, Zhongxing, Yin, Zhiwei, James, Clint A, Ruediger, Edward H, and Pearce, Bradley C

          PATENT:  US 2007078141  ISSUE DATE:  20070405

          APPLICATION: 2006-17538  PP: 67pp.

          ASSIGNEE:  (Bristol-Myers Squibb Company, USA

          View Data on the NIAID Therapeutics Website
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2.     60730   HIV-LS-373; SCIFINDER-HIV-4/23/2007

          Inhibitor of the folding of the HIV-1-protease as antiviral agent

          Broglia, Ricardo, Tiana, Guido, and Provasi, Davide

          PATENT:  US 2007072806  ISSUE DATE:  20070329

          APPLICATION: 2005-55852  PP: 17pp.

          ASSIGNEE:  (Universita' Degli Studi di Milano, Italy

          View Data on the NIAID Therapeutics Website
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3.     60731   HIV-LS-373; SCIFINDER-HIV-4/23/2007

          Synthetic polyvalent carbohydrates as components of HIV-1-blocking microbicides

          Wang, Lai-Xi, Wang, Jingsong, and Fouts, Timothy

          PATENT:  WO 2007033329  ISSUE DATE:  20070322

          APPLICATION: 2006  PP: 21pp.

          ASSIGNEE:  (University of Maryland Biotechnology Institute Off. of Research Admin./ Tech.Dev., USA

          View Data on the NIAID Therapeutics Website
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4.     60732   HIV-LS-373; SCIFINDER-HIV-4/23/2007

          Imidazo[1,2-a]pyridine compounds as chemokine receptor ligands and their preparation, pharmaceutical compositions and use in the treatment of HIV infection

          Gudmundsson, Kristjan and Boggs, Sharon Davis

          PATENT:  WO 2007027999  ISSUE DATE:  20070308

          APPLICATION: 2006  PP: 91pp.

          ASSIGNEE:  (Smithkline Beecham Corporation, USA

          View Data on the NIAID Therapeutics Website
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5.     60733   HIV-LS-373; WOS-HIV-4/30/2007

          Synthesis and Anti-Hiv-1 Activity of 1,3-Phenylene Bis-Uracil Analogues of Mkc-442

          Aly, Y. et al.

          Journal of Heterocyclic Chemistry 2007.  44(2): 381-387

          View Data on the NIAID Therapeutics Website
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          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000245494600016

6.     60734   HIV-LS-373; PUBMED-HIV-4/30/2007

          Drug design: New inhibitors for HIV-1 protease based on Nelfinavir as lead

          Perez, MA, Fernandes, PA, and Ramos, MJ

          J Mol Graph Model 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17459746&dopt=abstract


7.     60735   HIV-LS-373; PUBMED-HIV-4/30/2007

          De Novo Parallel Design, Synthesis and Evaluation of Inhibitors against the Reverse Transcriptase of Human Immunodeficiency Virus Type-1 and Drug-Resistant Variants

          Herschhorn, A, Lerman, L, Weitman, M, Gleenberg, IO, Nudelman, A, and Hizi, A

          J Med Chem 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17458947&dopt=abstract

8.     60736   HIV-LS-373; PUBMED-HIV-4/30/2007

          New AZT Analogues Having 5'-Alkylsulfonyl Groups: Synthesis and Anti-HIV Activity

          Al-Masoudi, NA, Al-Soud, YA, Ali, IA, Schuppler, T, Pannecouque, C, and De Clercq, E

          Nucleosides Nucleotides Nucleic Acids 2007.  26(3): 223-230

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17454731&dopt=abstract

9.     60737   HIV-LS-373; PUBMED-HIV-4/30/2007

          HIV protease inhibitors modulate apoptosis signaling in vitro and in vivo

          Vlahakis, SR, Bennett, SA, Whitehead, SN, and Badley, AD

          Apoptosis 2007.  12(5): 969-77

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17453162&dopt=abstract

10.   60738   HIV-LS-373; PUBMED-HIV-4/30/2007

          Heparin-mimicking sulfonic acid polymers as multitarget inhibitors of HIV-1 Tat and gp120 proteins

          Bugatti, A, Urbinati, C, Ravelli, C, De Clercq, E, Liekens, S, and Rusnati, M

          Antimicrob Agents Chemother 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17452490&dopt=abstract

11.   60739   HIV-LS-373; PUBMED-HIV-4/30/2007

          Structure-based identification of small molecule compounds targeting cell cyclophilin A with anti-HIV-1 activity

          Chen, S, Zhao, X, Tan, J, Lu, H, Qi, Z, Huang, Q, Zeng, X, Zhang, M, Jiang, S, Jiang, H, and Yu, L

          Eur J Pharmacol 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17449029&dopt=abstract


12.   60740   HIV-LS-373; PUBMED-HIV-4/30/2007

          Synthesis and evaluation of 2'-substituted cyclobutyl nucleosides and nucleotides as potential anti-HIV agents

          Li, Y, Mao, S, Hager, MW, Becnel, KD, Schinazi, RF, and Liotta, DC

          Bioorg Med Chem Lett 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17434736&dopt=abstract

13.   60741   HIV-LS-373; PUBMED-HIV-4/30/2007

          The Novel Fold of Scytovirin Reveals a New Twist For Antiviral Entry Inhibitors

          McFeeters, RL, Xiong, C, O'keefe, BR, Bokesch, HR, McMahon, JB, Ratner, DM, Castelli, R, Seeberger, PH, and Byrd, RA

          J Mol Biol 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17434526&dopt=abstract

14.   60742   HIV-LS-373; PUBMED-HIV-4/30/2007

          Tipranavir: a new protease inhibitor for the treatment of antiretroviral-experienced HIV-infected patients

          de Mendoza, C, Morello, J, Garcia-Gasco, P, Rodriguez-Novoa, S, and Soriano, V

          Expert Opin Pharmacother 2007.  8(6): 839-850

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17425479&dopt=abstract

15.   60743   HIV-LS-373; PUBMED-HIV-4/30/2007

          Biochemical Studies on the Mechanism of HIV-1 Reverse Transcriptase Resistance to 1-({beta}-D-Dioxolane)thymine Triphosphate

          Lennerstrand, J, Chu, CK, and Schinazi, RF

          Antimicrob Agents Chemother 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17403997&dopt=abstract

16.   60744   HIV-LS-373; PUBMED-HIV-4/30/2007

          Interaction between HIV-1 Rev and Integrase proteins: A basis for the development of anti-HIV peptides

          Rosenbluh, J, Hayouka, Z, Loya, S, Levin, A, Armon-Omer, A, Britan, E, Hizi, A, Kotler, M, Friedler, A, and Loyter, A

          J Biol Chem 2007.

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17403681&dopt=abstract


17.   60745   HIV-LS-373; PUBMED-HIV-4/30/2007

          Progesterone Inhibits HIV-1 Replication in Human Trophoblast Cells through Inhibition of Autocrine Tumor Necrosis Factor Secretion

          Diaz Munoz, L, Serramia, MJ, Fresno, M, and Munoz-Fernandez, MA

          J Infect Dis 2007.  195(9): 1294-302

          View Data on the NIAID Therapeutics Website
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          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17396998&dopt=abstract