ONLINE DATABASE SEARCH - HIV-LS-371-MEMO

 

1.     60537   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          Preparation of heterocyclic phenoxy compounds as HIV reverse transcriptase inhibitors

          Saggar, Sandeep A, Sisko, John T, Tucker, Thomas J, Tynebor, Robert M, Su, Dai-Shi, and Anthony, Neville J

          PATENT:  US 2007021442  ISSUE DATE:  20070125

          APPLICATION: 2006-29133  PP: 72pp.

          ASSIGNEE:  (USA)

          View Data on the NIAID Therapeutics Website
HYPERLINK:

2.     60538   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          Drug interactions of tipranavir, a new HIV protease inhibitor

          Morello, Judit, Rodriguez-Novoa, Sonia, Jimenez-Nacher, Inmaculada, and Soriano, Vincent

          Drug Metabolism Letters 2007.  1(1): 81-84

          View Data on the NIAID Therapeutics Website
HYPERLINK:

3.     60539   HIV-LS-371; PUBMED-HIV-4/3/2007

          A new era in HIV treatment: the entry inhibitors

          Berger, DS

          Posit Aware 2005.  16(1): 51-3

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17390505&dopt=abstract

4.     60540   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          Design, synthesis, and antiviral evaluation of some 3'-carboxymethyl-3'-deoxyadenosine derivatives

          Shi, Houguang, Ke, Pucheng, and Peterson, Matt A

          Abstracts of Papers, 233rd ACS National Meeting, Chicago, IL, United States, March 25-29, 2007  2007.: ORGN-389

          View Data on the NIAID Therapeutics Website
HYPERLINK:

5.     60541   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          3'-Fluoro-2',3'-unsaturated carbocyclic nucleosides: Synthesis, anti-HIV activity and molecular modeling studies

          Wang, Jianing, Jin, Yunho, Rapp, Kimberly L, Schinazi, Raymond F, and Chu, CK

          Abstracts of Papers, 233rd ACS National Meeting, Chicago, IL, United States, March 25-29, 2007  2007.: MEDI-073

          View Data on the NIAID Therapeutics Website
HYPERLINK:

6.     60542   HIV-LS-371; PUBMED-HIV-4/3/2007

          Synthesis and Anti-HIV-1 Activity Evaluation of 5-Alkyl-2-alkylthio-6-(arylcarbonyl or alpha-cyanoarylmethyl)-3,4-dihydropyrimidin-4(3H)-ones as Novel Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

          Ji, L, Chen, FE, DeClercq, E, Balzarini, J, and Pannecouque, C

          J Med Chem 2007.

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17381078&dopt=abstract


7.     60543   HIV-LS-371; PUBMED-HIV-4/3/2007

          Newer tetracycline derivatives: Synthesis, anti-HIV, antimycobacterial activities and inhibition of HIV-1 integrase

          Sriram, D, Yogeeswari, P, Senchani, G, and Banerjee, D

          Bioorg Med Chem Lett 2007.  17(8): 2372-5

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17376679&dopt=abstract

8.     60544   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          Novel 2-chloro-8-arylthiomethyldipyridodiazepinone derivatives with activity against HIV-1 reverse transcriptase

          Khunnawutmanotham, Nisachon, Chimnoi, Nitirat, Saparpakorn, Patchareenart, Pungpo, Pornpan, Louisirirotchanakul, Suda, Hannongbua, Supa, and Techasakul, Supanna

          Molecules 2007.  12(2): 218-230

          View Data on the NIAID Therapeutics Website
HYPERLINK:

9.     60545   HIV-LS-371; PUBMED-HIV-4/3/2007

          d- and l-2',3'-Didehydro-2',3'-dideoxy-3'-fluoro-carbocyclic Nucleosides: Synthesis, Anti-HIV Activity and Mechanism of Resistance

          Wang, J, Jin, Y, Rapp, KL, Schinazi, RF, and Chu, CK

          J Med Chem 2007.

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17373782&dopt=abstract

10.   60546   HIV-LS-371; PUBMED-HIV-4/3/2007

          A NOVEL bis-TETRAHYDROFURANYLURETHANE-CONTAINING NONPEPTIDIC PROTEASE INHIBITOR (PI) GRL-98065 POTENT AGAINST MULTI-PI-RESISTANT HIV IN VITRO

          Amano, M, Koh, Y, Das, D, Li, J, Leschenko, S, Wang, YF, Boross, PI, Weber, IT, Ghosh, AK, and Mitsuya, H

          Antimicrob Agents Chemother 2007.

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17371811&dopt=abstract

11.   60547   HIV-LS-371; PUBMED-HIV-4/3/2007

          Protein Design of a Bacterially Expressed HIV-1 gp41 Fusion Inhibitor

          Deng, Y, Zheng, Q, Ketas, TJ, Moore, JP, and Lu, M

          Biochemistry 2007.

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17371053&dopt=abstract


12.   60548   HIV-LS-371; PUBMED-HIV-4/3/2007

          HIV-1 reverse transcriptase inhibitors

          El Safadi, Y,  Vivet-Boudou, V, and Marquet, R

          Appl Microbiol Biotechnol 2007.

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17370068&dopt=abstract

13.   60549   HIV-LS-371; PUBMED-HIV-4/3/2007

          Development of integrase inhibitors for treatment of AIDS: An overview

          Dubey, S, Satyanarayana, YD, and Lavania, H

          Eur J Med Chem  2007.

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17367896&dopt=abstract

14.   60550   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          The Vif accessory protein alters the cell cycle of human immunodeficiency virus type 1 infected cells

          Wang, Jiangfang, Shackelford, Jason M, Casella, Carolyn R, Shivers, Debra K, Rapaport, Eric L, Liu, Bindong, Yu, Xiao-Fang, and Finkel, Terri H

          Virology 2007.  359(2): 243-252

          View Data on the NIAID Therapeutics Website
HYPERLINK:

15.   60551   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          1,5-Naphthyridin-2(1H)-one derivative HIV integrase inhibitors, and use with other agents

          Johns, Brian A and Spaltenstein, Andrew

          PATENT:  WO 2007019130  ISSUE DATE:  20070215

          APPLICATION: 2006  PP: 47pp.

          ASSIGNEE:  (Smithkline Beecham Corporation, USA

          View Data on the NIAID Therapeutics Website
HYPERLINK:

16.   60552   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          2-oxonaphthyridine-3-carboxamides as HIV integrase inhibitors and their preparation and use in the prevention and treatment of HIV infection, AIDS and ARC

          Johns, Brian A and Spaltenstein, Andrew

          PATENT:  WO 2007019101  ISSUE DATE:  20070215

          APPLICATION: 2006  PP: 78pp.

          ASSIGNEE:  (Smithkline Beecham Corporation, USA

          View Data on the NIAID Therapeutics Website
HYPERLINK:

17.   60553   HIV-LS-371; PUBMED-HIV-4/3/2007

          Enzymatically Activated cycloSal-d4T-monophosphates: The Third Generation of cycloSal-Pronucleotides

          Gisch, N, Balzarini, J, and Meier, C

          J Med Chem 2007.  50(7): 1658-1667

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=17335187&dopt=abstract


18.   60554   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          Noninfectious papilloma virus-like particles inhibit HIV-1 replication: implications for immune control of HIV-1 infection by IL-27

          Mohamad Fakruddin, J, Lempicki, Richard A, Gorelick, Robert J, Yang, Jun, Adelsberger, Joseph W, Garcia-Pineres, Alfonso J, Pinto, Ligia A, Lane, HClifford, and Imamichi, Tomozumi

          Blood 2007.  109(5): 1841-1849

          View Data on the NIAID Therapeutics Website
HYPERLINK:

19.   60555   HIV-LS-371; WOS-HIV-3/25/2007

          1,2,3-Triazoles as peptide bond isosteres: synthesis and biological evaluation of cyclotetrapeptide mimics

          Bock, VD, Speijer, D, Hiemstra, H, and van Maarseveen, JH

          ORGANIC & BIOMOLECULAR CHEMISTRY 2007.  5(6): 971-975, 5

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000244703800014

20.   60556   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          naphthyridinecarboxamides as HIV integrase inhibitors and their preparation, pharmaceutical compositions and use in the treatment of HIV infections, AIDS and ARC

          Johns, Brian A

          PATENT:  WO 2007019098  ISSUE DATE:  20070215

          APPLICATION: 2006  PP: 132pp.

          ASSIGNEE:  (Smithkline Beecham Corporation, USA, Shionogi & Co. Ltd, and Kawasuji, Takashi

          View Data on the NIAID Therapeutics Website
HYPERLINK:

21.   60557   HIV-LS-371; SCIFINDER-HIV-3/26/2007

          Preparation of alanine phosphonate derivatives as antiviral agents

          Cai, Zhenhong R, Jabri, Salman Y, Jin, Haolun, Kim, Choung U, Metobo, Samuel E, Mish, Michael R, and Pastor, Richard M

          PATENT:  WO 2007014352  ISSUE DATE:  20070201

          APPLICATION: 2006  PP: 195pp.

          ASSIGNEE:  (Gilead Sciences, Inc. USA

          View Data on the NIAID Therapeutics Website
HYPERLINK:

22.   60558   HIV-LS-371; WOS-HIV-3/25/2007

          Inhibition of human immunodeficiency virus type-1 reverse transcriptase by a novel peptide derived from the viral integrase

          Gleenberg, IO, Herschhorn, A, Goldgur, Y, and Hizi, A

          ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS 2007.  458(2): 202-212, 11

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000244385000014

23.   60559   HIV-LS-371; WOS-HIV-3/25/2007

          Chemokine antagonists as therapeutics: Focus on HIV-1

          Tsibris, AMN and Kuritzkes, DR

          ANNUAL REVIEW OF MEDICINE 2007.  58: 445-459, 15

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000244461500030

24.   60560   HIV-LS-371; WOS-HIV-3/25/2007

          Elimination of HIV-1 infection by treatment with a doxorubicin-conjugated anti-envelope antibody

          Johansson, S, Goldenberg, DM, Griffiths, GL, Wahren, B, and Hinkula, J

          AIDS 2006.  20 (15): 1911-1915, 5

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000244509800002

25.   60561   HIV-LS-371; WOS-HIV-3/25/2007

          Synthesis of guanidinoxylopyranosides and their anti-HIV PR activity

          Cao, LH and Lian, ZB

          ACTA CHIMICA SINICA 2007.  65(4): 349-354, 6

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000244500200013

26.   60562   HIV-LS-371; WOS-HIV-4/2/2007

          Inhibition of HIV-1 integrase by modified oligonucleotides: Optimization of the inhibitor structure

          Prikazchikova, TA, Volkov, EM, Zubin, EM, Romanova, EA, and Gottikh, MB

          MOLECULAR BIOLOGY 2007.  41(1): 118-125, 8

          View Data on the NIAID Therapeutics Website
HYPERLINK:

          http://publishorperish.nih.gov/Gateway.cgi?KeyUT=000244508100016